SCHEMBL7743898

SCHEMBL7743898

N#Cc1ccc(CC(C(=O)O)c2cnc[nH]2)cc1F.[LiH]

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 17/20 0.62
CPA1 P15085 1/20 0.57
CPB1 P15086 5/20 0.54
DAO P14920 1/20 0.41
CYP19A1 P11511 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lithium Ion SCHEMBL7743896 0.88 CPB2 (0.50) CPB2CPA1CPB1DAOCYP19A1
SCHEMBL7743300 0.86 CPB2 (0.48) CPB2CPA1CPB1DAO
SCHEMBL7053727 0.80 CPA1 (0.71) CPB2CPA1CPB1CYP19A1
Hydrochloric Acid SCHEMBL8495732 0.79 CPA1 (0.69) CPB2CPA1CPB1CYP19A1
SCHEMBL8865742 0.78 CPA1 (0.76) CPB2CPA1CPB1CYP19A1
SCHEMBL7704747 0.76 CACNA1H (0.40) CPB2DAOCYP19A1
Hydrochloric Acid SCHEMBL8763045 0.73 CPA1 (0.71) CPB2CPA1CPB1
SCHEMBL25220822 0.73 TRPV4 (0.45) DAO
Hydrochloric Acid SCHEMBL8763128 0.73 CPA1 (0.97) CPB2CPA1CPB1
SCHEMBL2322118 0.72 SLC7A5 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091736-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2001-10-24 EP disclosed
EP-1091736-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-18 EP disclosed
WO-2000001382-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed