SCHEMBL7744588

SCHEMBL7744588

CCCN1C(=O)C(C(C(N)=O)c2ccc(C(F)(F)F)cc2C(F)(F)F)N=C(C2CC2)c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 10/20 0.44
BDKRB1 P46663 6/20 0.40
KCNH2 Q12809 1/20 0.39
NOTCH1 P46531 3/20 0.36
NOTCH3 Q9UM47 2/20 0.36
RBPJ Q06330 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744126 0.78 CCKBR (0.42) CCKBRBDKRB1KCNH2
SCHEMBL7743998 0.73 KCNH2 (0.61) CCKBRBDKRB1KCNH2
SCHEMBL7738908 0.73 KCNH2 (0.45) CCKBRKCNH2NOTCH1NOTCH3RBPJ
SCHEMBL7744128 0.69 KCNH2 (0.52) CCKBRKCNH2
SCHEMBL7744120 0.68 KCNH2 (0.36) CCKBRBDKRB1KCNH2
SCHEMBL7743995 0.68 KCNH2 (0.36) CCKBRBDKRB1KCNH2
SCHEMBL8620108 0.67 KCNH2 (0.77) CCKBRKCNH2
SCHEMBL7744124 0.67 KCNH2 (0.55) CCKBRKCNH2
SCHEMBL7744000 0.67 KCNH2 (0.55) CCKBRKCNH2
SCHEMBL9214723 0.67 BDKRB1 (0.49) CCKBRBDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001010216-A1 ANTIARRHYTHMIC COMPOUNDS MERCK & CO., INC. (US) 2001-02-15 WO disclosed