SCHEMBL7744780

SCHEMBL7744780

CCOC(=O)CCC(C#N)(CCC(=O)OCC)c1ccc(F)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.35
BRCA1 P38398 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 1/20 0.35
CYP4F2 P78329 2/20 0.35
CYP4A11 Q02928 2/20 0.35
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HPGD P15428 2/20 0.34
TSHR P16473 1/20 0.34
POLB P06746 1/20 0.34
ESR1 P03372 1/20 0.34
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KCNN4 O15554 1/20 0.33
NLRP3 Q96P20 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744784 0.95 SMN1; SMN2 (0.34) CASP1HSD17B10ALDH1A1MEN1BRCA1
SCHEMBL11826001 0.88 CASP1 (0.47) CASP1HSD17B10ALDH1A1LMNAHPGD
SCHEMBL7744791 0.87 HSD17B10 (0.41) CASP1HSD17B10ALDH1A1KMT2AMAPT
SCHEMBL6997987 0.87 MAPT (0.36) HSD17B10ALDH1A1MAPTHPGDTSHR
SCHEMBL7749356 0.84 MAPT (0.38) CASP1HSD17B10ALDH1A1MEN1KMT2A
SCHEMBL7744793 0.82 HSD17B10 (0.38) CASP1HSD17B10ALDH1A1KMT2AMAPT
SCHEMBL7750623 0.82 SMN1; SMN2 (0.39) CASP1HSD17B10ALDH1A1KMT2AMAPT
SCHEMBL7752046 0.81 RORC (0.36) CASP1HSD17B10ALDH1A1KMT2AMAPT
SCHEMBL11819756 0.81 ESR1 (0.48) CASP1HSD17B10ALDH1A1MEN1KMT2A
SCHEMBL7749384 0.81 KCNN4 (0.41) CASP1HSD17B10ALDH1A1TSHRESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242607-B1 SUCH AS 4-CYANO-4-(3,4-DICHLOROPHENYL)HEPTANEDIOIC ACID USED AS ANTAGONISTS OF NEUROKININES SANOFI-SYNTHELABO (FR) 2001-06-05 US disclosed
US-6008360-A Substituted 3-aryl-3-carboxyalkyl glutaramides, method for preparing same by 4-arylo-4-cyanoheptane dicarboxylic acid cyclisation, and use thereof for preparing 3-aryl-3-hydroxyalkylpiperidines SANOFI-SYNTHELABO (FR) 1999-12-28 US disclosed