SCHEMBL7744784

SCHEMBL7744784

CCOC(=O)CCC(C#N)(CCC(=O)O)c1ccc(F)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 4/20 0.34
HSD17B10 Q99714 2/20 0.34
CASP1 P29466 1/20 0.34
POLB P06746 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KCNN4 O15554 1/20 0.33
BRCA1 P38398 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPT P10636 1/20 0.33
ESR1 P03372 1/20 0.33
CYP3A4 P08684 1/20 0.33
ESR2 Q92731 1/20 0.33
FFAR1 O14842 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
LMNA P02545 1/20 0.32
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744780 0.95 CASP1 (0.36) SMN1; SMN2ALDH1A1HSD17B10CASP1POLB
SCHEMBL7744793 0.88 HSD17B10 (0.38) ALDH1A1HSD17B10CASP1KMT2AKCNN4
SCHEMBL7749384 0.88 KCNN4 (0.41) ALDH1A1HSD17B10CASP1KCNN4ESR1
SCHEMBL7749357 0.85 MAPT (0.35) SMN1; SMN2ALDH1A1HSD17B10CASP1MEN1
SCHEMBL7750624 0.84 SMN1; SMN2 (0.36) SMN1; SMN2ALDH1A1HSD17B10CASP1POLB
SCHEMBL11826001 0.84 CASP1 (0.47) ALDH1A1HSD17B10CASP1KDM4ELMNA
SCHEMBL4439878 0.83 MEN1 (0.36) SMN1; SMN2ALDH1A1HSD17B10POLBMEN1
SCHEMBL4431094 0.83 KYAT1 (0.40) SMN1; SMN2ALDH1A1POLBMEN1KMT2A
SCHEMBL734031 0.83 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1POLBMEN1KMT2A
SCHEMBL6997987 0.83 MAPT (0.36) ALDH1A1HSD17B10KCNN4KDM4EALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242607-B1 SUCH AS 4-CYANO-4-(3,4-DICHLOROPHENYL)HEPTANEDIOIC ACID USED AS ANTAGONISTS OF NEUROKININES SANOFI-SYNTHELABO (FR) 2001-06-05 US disclosed
US-6008360-A Substituted 3-aryl-3-carboxyalkyl glutaramides, method for preparing same by 4-arylo-4-cyanoheptane dicarboxylic acid cyclisation, and use thereof for preparing 3-aryl-3-hydroxyalkylpiperidines SANOFI-SYNTHELABO (FR) 1999-12-28 US disclosed