SCHEMBL7749356

SCHEMBL7749356

CC(C)OC(=O)CCC(C#N)(CCC(=O)OC(C)C)c1ccc(F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.38
CASP1 P29466 2/20 0.36
HSD17B10 Q99714 2/20 0.36
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ESR1 P03372 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KCNN4 O15554 1/20 0.33
TSHR P16473 1/20 0.33
CETP P11597 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7749357 0.95 MAPT (0.35) MAPTCASP1HSD17B10GAASMN1; SMN2
SCHEMBL7744791 0.86 HSD17B10 (0.41) MAPTCASP1HSD17B10GAAKMT2A
SCHEMBL11832348 0.84 MAPT (0.40) MAPTMEN1KMT2AKCNN4TSHR
SCHEMBL7744780 0.84 CASP1 (0.36) MAPTCASP1HSD17B10GAASMN1; SMN2
SCHEMBL7744793 0.81 HSD17B10 (0.38) MAPTCASP1HSD17B10GAAESR1
SCHEMBL7752046 0.80 RORC (0.36) MAPTCASP1HSD17B10GAAKMT2A
SCHEMBL7749384 0.80 KCNN4 (0.41) CASP1HSD17B10ESR1KCNN4TSHR
SCHEMBL7744784 0.80 SMN1; SMN2 (0.34) MAPTCASP1HSD17B10GAASMN1; SMN2
SCHEMBL11820141 0.77 KDM4E (0.38) MAPTCASP1HSD17B10GAASMN1; SMN2
SCHEMBL7752049 0.76 CASP1 (0.34) MAPTCASP1HSD17B10GAAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242607-B1 SUCH AS 4-CYANO-4-(3,4-DICHLOROPHENYL)HEPTANEDIOIC ACID USED AS ANTAGONISTS OF NEUROKININES SANOFI-SYNTHELABO (FR) 2001-06-05 US disclosed
US-6008360-A Substituted 3-aryl-3-carboxyalkyl glutaramides, method for preparing same by 4-arylo-4-cyanoheptane dicarboxylic acid cyclisation, and use thereof for preparing 3-aryl-3-hydroxyalkylpiperidines SANOFI-SYNTHELABO (FR) 1999-12-28 US disclosed
US-3979444-A CENTRAL NERVOUS SYSTEM DEPRESSANTS, HYPOTENSIVES THE UPJOHN COMPANY (US) 1976-09-07 US disclosed