SCHEMBL7745264

SCHEMBL7745264

COC(=O)CCOc1c[c]c(F)cc1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TP53 P04637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ALDH1A1 P00352 4/20 0.41
HPGD P15428 3/20 0.41
TSHR P16473 1/20 0.41
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
CYP1A2 P05177 1/20 0.38
GLA P06280 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
AR P10275 1/20 0.37
FFAR1 O14842 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595259 0.87 AR (0.48) NPC1RAB9ATP53HSD17B10ALDH1A1
SCHEMBL8807177 0.80 MAPT (0.50) NPC1RAB9AALDH1A1HPGDTSHR
SCHEMBL5843410 0.79 ALDH1A1 (0.38) NPC1RAB9ATP53HSD17B10ALDH1A1
SCHEMBL5841619 0.77 NLRP3 (0.43) HSD17B10ALDH1A1HPGDTSHRMAPT
SCHEMBL5843345 0.74 ALDH1A1 (0.44) ALDH1A1KDM4EAR
SCHEMBL5844399 0.73 ALOX5AP (0.32)
SCHEMBL5842046 0.73 ALDH1A1 (0.35) HSD17B10ALDH1A1HPGDTSHRKDM4E
SCHEMBL6595260 0.73 MAPT (0.56) NPC1RAB9ATP53HSD17B10ALDH1A1
SCHEMBL8894491 0.72 ALDH1A1 (0.33) ALDH1A1HPGDTSHRAR
SCHEMBL4845134 0.72 ALDH1A1 (0.72) NPC1RAB9ATP53HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001009087-A1 SUBSTITUTED ARYLHYDRAZONE CARBOXYLIC ACID DERIVATIVES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2001-02-08 WO disclosed
EP-1070055-A1 SUBSTITUTED PHENYL PYRIDAZINONES Bayer Aktiengesellschaft (DE) 2001-01-24 EP disclosed
WO-2000008000-A1 USE OF SUBSTITUTED TRIAZINONES AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2000-02-17 WO disclosed
WO-1999052878-A1 SUBSTITUTED PHENYL PYRIDAZINONES BAYER AKTIENGESELLSCHAFT (DE) 1999-10-21 WO disclosed
WO-1997005117-A1 SUBSTITUTED 1-PHENYLURACIL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-02-13 WO disclosed