SCHEMBL7745986

SCHEMBL7745986

Nc1c(Br)cc(S(=O)(=O)C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
CYP3A4 P08684 1/20 0.51
PTPN1 P18031 1/20 0.47
CTSB P07858 1/20 0.46
L3MBTL1 Q9Y468 3/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.43
MAPK1 P28482 1/20 0.43
RECQL P46063 1/20 0.43
CA1 P00915 6/20 0.43
CA2 P00918 6/20 0.43
CA9 Q16790 6/20 0.43
CA12 O43570 4/20 0.43
ALDH3A1 P30838 1/20 0.42
CA3 P07451 1/20 0.42
EPAS1 Q99814 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
VCAM1 P19320 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7752783 0.83 ALDH1A1 (0.46) ALDH1A1CYP3A4PTPN1L3MBTL1LMNA
SCHEMBL999002 0.83 CA2 (0.59) ALDH1A1LMNAMAPTCA1CA2
SCHEMBL7769730 0.82 ALDH1A1 (0.56) ALDH1A1CYP3A4CTSBL3MBTL1CA1
SCHEMBL5840961 0.82 CA1 (0.64) ALDH1A1CYP3A4CTSBL3MBTL1MAPT
SCHEMBL9186437 0.81 PTPN1 (0.56) ALDH1A1PTPN1L3MBTL1LMNAMAPT
SCHEMBL31646963 0.79 ALDH1A1 (0.56) ALDH1A1CYP3A4CTSBL3MBTL1CA1
SCHEMBL5840098 0.79 ALDH1A1 (0.56) ALDH1A1CYP3A4CTSBL3MBTL1CA1
SCHEMBL7750641 0.78 ALDH1A1 (0.55) ALDH1A1LMNACA1CA2CA9
SCHEMBL5786092 0.78 ALDH1A1 (0.64) ALDH1A1CYP3A4PTPN1L3MBTL1LMNA
SCHEMBL31646617 0.76 ALDH1A1 (0.49) ALDH1A1CYP3A4CTSBL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0597304-B1 Use of substituted benzimidazoles for combating parasitic protozoas BAYER AG (DE) 2001-01-10 EP disclosed
US-5877195-A INSECTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1999-03-02 US disclosed
US-5863933-A NEMATOCIDES, PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1999-01-26 US disclosed
EP-0596358-B1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1998-10-28 EP disclosed
US-5656649-A PESTICIDE, INSECTICIDES, NEMATOCIDE BAYER AKTIENGESELLSCHAFT (DE) 1997-08-12 US disclosed
US-5585395-A INSECTICIDES, MITICIDES, FUNGICIDES, HERBICIDES, PLANT GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1996-12-17 US disclosed
US-5484953-A CHEMICAL INTERMEDIATES FOR BENZIMIDAZOLES FOR INSECTICIDES OR NEMATOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-01-16 US disclosed
US-5482956-A ANTIPROTOZOA AGENTS FOR ANIMALS OR INSECTS BAYER AKTIENGESELLSCHAFT (DE) 1996-01-09 US disclosed
EP-0597304-A1 Use of substituted benzimidazoles BAYER AG (DE) 1994-05-18 EP disclosed
EP-0596358-A1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1994-05-11 EP disclosed