SCHEMBL7746219

SCHEMBL7746219

CCCCC(=O)Nc1c(NCc2ccc(C(=O)O)cc2)ncnc1OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.44
POLB P06746 3/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
BDKRB1 P46663 1/20 0.43
EGFR P00533 3/20 0.42
TDP1 Q9NUW8 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HDAC3 O15379 2/20 0.40
ERBB2 P04626 1/20 0.40
KDR P35968 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7751822 0.90 BDKRB1 (0.46) POLBBDKRB1EGFRTDP1ALDH1A1
SCHEMBL7752068 0.88 BDKRB1 (0.44) BDKRB1EGFRALDH1A1HDAC3ERBB2
SCHEMBL7753196 0.84 ALDH1A1 (0.46) POLBBDKRB1EGFRTDP1ALDH1A1
SCHEMBL7753157 0.83 BDKRB1 (0.53) POLBMAPTBDKRB1EGFRTDP1
SCHEMBL7752026 0.82 SMN1; SMN2 (0.47) POLBBDKRB1EGFR
SCHEMBL7750841 0.80 EGFR (0.52) POLBBDKRB1EGFRALDH1A1HDAC3
SCHEMBL7753138 0.79 LTB4R2 (0.40) POLBBDKRB1EGFRTDP1ALDH1A1
SCHEMBL7746182 0.78 BDKRB1 (0.49) POLBMAPTBDKRB1EGFRTDP1
SCHEMBL7750817 0.75 ALDH1A1 (0.52) POLBMAPTBDKRB1EGFRALDH1A1
SCHEMBL7746181 0.74 BDKRB1 (0.48) MAPTBDKRB1EGFRALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686631-B1 Pyrimidine derivatives and pharmaceutical compositions KUREHA CHEMICAL IND CO LTD (JP) 2001-01-17 EP disclosed
EP-0686631-A1 Pyrimidine derivatives and pharmaceutical composition Kureha Chemical Industry Co., Ltd. (JP) 1995-12-13 EP disclosed