SCHEMBL7748936

SCHEMBL7748936

O=C1Nc2ccc(F)cc2C2(CCN(CCCCCN3C(=O)OC[C@@H]3c3ccc(F)c(F)c3)CC2)O1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.43
PLD2 O14939 2/20 0.37
PLD1 Q13393 2/20 0.37
ADRA1A P35348 12/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ADRA1D P25100 11/20 0.36
ADRA1B P35368 11/20 0.36
TDP1 Q9NUW8 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
HRH1 P35367 1/20 0.35
HTR7 P34969 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7743435 0.93 CCR2 (0.39) CCR2ADRA1ATP53CYP3A4MAPT
SCHEMBL7743434 0.93 CCR2 (0.39) CCR2ADRA1ATP53CYP3A4MAPT
SCHEMBL7747425 0.77 ADRA1A (0.49) ADRA1AADRA1DADRA1BHRH1
SCHEMBL7675111 0.77 ADRA1D (0.43) ADRA1AADRA1DADRA1B
SCHEMBL7679189 0.77 ADRA1D (0.43) ADRA1AADRA1DADRA1B
SCHEMBL7679689 0.77 ADRA1D (0.43) ADRA1AADRA1DADRA1B
SCHEMBL4999332 0.73 CCR2 (0.49) CCR2PLD2PLD1ADRA1ATP53
SCHEMBL4999331 0.73 CCR2 (0.49) CCR2PLD2PLD1ADRA1ATP53
SCHEMBL5663717 0.72 MTOR (0.34) ADRA1AADRA1DADRA1B
SCHEMBL7678845 0.72 MTOR (0.34) ADRA1AADRA1DADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001022919-A2 SPIRO[BICYCLIC -AZACYCLOALKYL AND -CYCLOALKYL] DERIVATIVES AND USES THEREOF MERCK & CO., INC. (US) 2001-04-05 WO claimed