SCHEMBL7749030

SCHEMBL7749030

CN1C(=O)OC2(CCN(CCCCN3C(=O)c4ccccc4S3(=O)=O)CC2)c2cc(Cl)ccc21

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.55
DRD4 P21917 3/20 0.55
DRD5 P21918 3/20 0.55
DRD3 P35462 3/20 0.55
HTR1A P08908 11/20 0.54
HTR2A P28223 11/20 0.54
HTR7 P34969 11/20 0.54
HTR6 P50406 11/20 0.54
ADRA1D P25100 1/20 0.51
ADRA1A P35348 1/20 0.51
ADRA1B P35368 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7748894 0.93 ADRA1D (0.55) DRD2DRD4DRD5DRD3HTR1A
SCHEMBL7656937 0.70 HRH1 (0.45)
SCHEMBL8804131 0.69 DRD2 (0.56) DRD2DRD4DRD5DRD3HTR1A
SCHEMBL7815142 0.69 DRD2 (0.71) DRD2DRD4DRD5DRD3HTR1A
Du 125530 SCHEMBL29403202 0.69 HTR1A (0.68) DRD2DRD4DRD5DRD3HTR1A
Du 125530 SCHEMBL1082516 0.69 HTR1A (0.68) DRD2DRD4DRD5DRD3HTR1A
SCHEMBL7822015 0.68 DRD2 (0.67) DRD2DRD4DRD5DRD3HTR1A
SCHEMBL7820656 0.68 HTR1A (0.67) DRD2DRD4DRD5DRD3HTR1A
Du 125530 SCHEMBL6063602 0.68 HTR1A (0.67) DRD2DRD4DRD5DRD3HTR1A
SCHEMBL7656122 0.68 HRH1 (0.43) ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001022919-A2 SPIRO[BICYCLIC -AZACYCLOALKYL AND -CYCLOALKYL] DERIVATIVES AND USES THEREOF MERCK & CO., INC. (US) 2001-04-05 WO disclosed