Ly-255283

Ly-255283

SCHEMBL7749547

CCc1cc(C(C)=O)c(O)cc1OCCCCCC(C)(C)c1nn[nH]n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 16/20 1.00
LTB4R Q15722 5/20 1.00
LTB4R2 Q9NPC1 5/20 1.00
MEN1 O00255 1/20 1.00
ALDH1A1 P00352 1/20 1.00
CYP3A4 P08684 1/20 1.00
THRB P10828 1/20 1.00
HPGD P15428 1/20 1.00
ALOX15 P16050 1/20 1.00
TSHR P16473 1/20 1.00
HTR2B P41595 1/20 1.00
KMT2A Q03164 1/20 1.00
HSD17B10 Q99714 1/20 1.00
SIGMAR1 Q99720 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9431167 0.89 NR1H4 (1.00) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL7751099 0.86 LTB4R (1.00) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL8652398 0.86 LTB4R (0.85) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL8651177 0.85 LTB4R (0.83) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL8653365 0.85 LTB4R (0.86) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL8655402 0.85 LTB4R (0.98) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL9430782 0.85 LTB4R (0.98) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL9431492 0.85 LTB4R (0.86) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL9431503 0.85 LTB4R (0.86) NR1H4LTB4RLTB4R2MEN1ALDH1A1
SCHEMBL9430787 0.85 LTB4R (0.98) NR1H4LTB4RLTB4R2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001034199-A2 ONCOLYTIC COMBINATIONS FOR THE TREATMENT OF CANCER ELI LILLY AND COMPANY (US) 2001-05-17 WO claimed
US-9861601-B2 Treatment of pulmonary arterial hypertension with leukotriene inhibitors THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2018-01-09 US disclosed
US-20160193168-A1 Treatment of Pulmonary Arterial Hypertension with Leukotriene Inhibitors THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2016-07-07 US disclosed
US-20160193168-A1 Treatment of Pulmonary Arterial Hypertension with Leukotriene Inhibitors THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2016-07-07 US disclosed
US-20160166508-A1 Method and Composition for Treating Inflammatory Disorders MEDA AB (SE) 2016-06-16 US disclosed
US-20160166508-A1 Method and Composition for Treating Inflammatory Disorders MEDA AB (SE) 2016-06-16 US disclosed
US-9233089-B2 Treatment of pulmonary hypertension with leukotriene inhibitors THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2016-01-12 US disclosed
US-9233089-B2 Treatment of pulmonary hypertension with leukotriene inhibitors THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2016-01-12 US disclosed
EP-2827849-A1 TREATMENT OF PULMONARY HYPERTENSION WITH LEUKOTRIENE INHIBITORS The Board Of Trustees Of The University Of the Leland Stanford Junior University (US) 2015-01-28 EP disclosed
WO-2013142369-A1 TREATMENT OF PULMONARY HYPERTENSION WITH LEUKOTRIENE INHIBITORS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-09-26 WO disclosed
WO-2013142369-A1 TREATMENT OF PULMONARY HYPERTENSION WITH LEUKOTRIENE INHIBITORS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-09-26 WO disclosed
US-20130251787-A1 Treatment of Pulmonary Hypertension with Leukotriene Inhibitors THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-09-26 US disclosed
US-20130251787-A1 Treatment of Pulmonary Hypertension with Leukotriene Inhibitors THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-09-26 US disclosed
US-20090220583-A1 Method and composition for treating inflammatory disorders MEDA AB (SE) 2009-09-03 US disclosed
US-20090220583-A1 Method and composition for treating inflammatory disorders MEDA AB (SE) 2009-09-03 US disclosed
US-20080081835-A1 Use of Ltb4 Inhibitors for the Treatment of B-Cell Leukemias and Lymphomas BIOLIPOX AB (SE) 2008-04-03 US disclosed
US-20080081835-A1 Use of Ltb4 Inhibitors for the Treatment of B-Cell Leukemias and Lymphomas BIOLIPOX AB (SE) 2008-04-03 US disclosed
WO-2001034134-A2 ONCOLYTIC COMBINATIONS FOR THE TREATMENT OF CANCER ELI LILLY AND COMPANY (US) 2001-05-17 WO disclosed
WO-2001034133-A2 ONCOLYTIC COMBINATIONS FOR THE TREATMENT OF CANCER ELI LILLY AND COMPANY (US) 2001-05-17 WO disclosed
WO-2001034199-A2 ONCOLYTIC COMBINATIONS FOR THE TREATMENT OF CANCER ELI LILLY AND COMPANY (US) 2001-05-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130251787-A1 Treatment of Pulmonary Hypertension with Leukotriene Inhibitors LTA4H, LTB4R2, LTB4R NR1H4 1045/4885LTB4R 3/4885LTB4R2 2/4885
US-20090220583-A1 Method and composition for treating inflammatory disorders LIPA, HRH2, HRH1 NR1H4 97/4885LTB4R 8/4885LTB4R2 7/4885
US-20160193168-A1 Treatment of Pulmonary Arterial Hypertension with Leukotriene Inhibitors LTA4H, LTB4R2, LTB4R NR1H4 1508/4885LTB4R 3/4885LTB4R2 2/4885
US-20160166508-A1 Method and Composition for Treating Inflammatory Disorders LIPA, HRH2, HRH1 NR1H4 97/4885LTB4R 8/4885LTB4R2 7/4885
US-20080081835-A1 Use of Ltb4 Inhibitors for the Treatment of B-Cell Leukemias and Lymphomas LTB4R, LTA4H, LTA NR1H4 637/4885LTB4R 1/4885LTB4R2 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.