SCHEMBL7749803

SCHEMBL7749803

O=CC1=CCCc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.43
MAOB P27338 2/20 0.39
MAOA P21397 2/20 0.39
CYP2A6 P11509 1/20 0.39
PDPK1 O15530 1/20 0.37
PARP1 P09874 1/20 0.37
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
MAPT P10636 2/20 0.35
PKM P14618 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
MIF P14174 2/20 0.34
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
SRD5A1 P18405 1/20 0.33
SRD5A2 P31213 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29648452 1.00 CES1 (0.43) CES1MAOBMAOACYP2A6PDPK1
SCHEMBL2675857 0.82 ALOX5 (0.38) CES1MAOBMAOACYP2A6PDPK1
SCHEMBL2863342 0.81 HTR6 (0.42) CES1MAOBMAOACYP2A6PDPK1
SCHEMBL15780617 0.80 CES1 (0.39) CES1MAOBMAOACYP2A6PDPK1
SCHEMBL5327197 0.78 MEN1 (0.36) MAOBMAOACYP2A6L3MBTL1
SCHEMBL2526007 0.77 CES1 (0.48) CES1MAOBMAOACYP2A6PDPK1
SCHEMBL19775784 0.72 CES1 (0.39) CES1MAOBMAOACYP2A6PDPK1
SCHEMBL2674629 0.72 SIGMAR1 (0.43) CES1MAOBMAOACYP2A6PDPK1
SCHEMBL28780467 0.71 PARP10 (0.44) CYP2A6PARP10PARP11
SCHEMBL22682127 0.70 AR (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114605314-B Indene derivative and application thereof 上海八亿时空先进材料有限公司 2024-04-02 CN disclosed
WO-2023161857-A1 BIFUNCTIONAL CYTOKINE COMPOSITIONS BRIGHT PEAK THERAPEUTICS AG (CH) 2023-08-31 WO disclosed
CN-114605314-A Indene derivative and application thereof 上海八亿时空先进材料有限公司 2022-06-10 CN disclosed
WO-2001042181-A1 BENZYL TETRALINS, FORMULATIONS AND USES THEREOF UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 2001-06-14 WO disclosed
EP-0540697-A1 NOVEL SULFONYLUREAS Novartis AG (CH) 1993-05-12 EP disclosed
EP-0281283-B1 HETEROCYCLIC COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-10 EP disclosed
US-4910212-A Containing 1,2,4-triazole or imidazole ring IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-03-20 US disclosed
EP-0281283-A1 Heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-09-07 EP disclosed