SCHEMBL7750587

SCHEMBL7750587

CC(NNC(N)=O)Oc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.46
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
GLA P06280 1/20 0.44
TDP1 Q9NUW8 2/20 0.42
TSHR P16473 2/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
GAA P10253 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 2/20 0.41
HTT P42858 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19544761 0.74 SLC6A4 (0.42) POLBMTNR1AMTNR1BMEN1KMT2A
SCHEMBL11384019 0.73 MTNR1A (0.57) MTNR1AMTNR1BMEN1KMT2AGAA
SCHEMBL8652167 0.73 ALDH1A1 (0.47) POLBTDP1MEN1KMT2AALDH1A1
SCHEMBL27671316 0.72 POLB (0.60) POLBTDP1TSHRMEN1KMT2A
SCHEMBL1328578 0.72 GAA (0.56) POLBMTNR1AMTNR1BTDP1TSHR
SCHEMBL1684925 0.72 BCAT2 (0.47) KMT2AGAAALDH1A1LMNACYP1A2
SCHEMBL6804593 0.71 ALDH1A1 (0.41) POLBMTNR1AMTNR1BTSHRMEN1
SCHEMBL17046780 0.71 POLB (0.41) POLBMTNR1AMTNR1BMEN1KMT2A
SCHEMBL7979605 0.71 MTNR1A (0.47) POLBMTNR1AMTNR1BTDP1TSHR
SCHEMBL11402564 0.71 MAOA (0.52) POLBMTNR1AMTNR1BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0568437-B1 Antidepressant 3-Halophenylpiperazinyl-propyl Derivatives of Substituted Triazolones and Triazoldiones BRISTOL MYERS SQUIBB CO (US) 2001-02-21 EP disclosed
EP-0568437-A1 Antidepressant 3-Halophenylpiperazinyl-propyl Derivatives of Substituted Triazolones and Triazoldiones Bristol-Myers Squibb Company (US) 1993-11-03 EP disclosed
US-5256664-A Antidepressant 3-halophenylpiperazinylpropyl derivatives of substituted triazolones and triazoldiones BRISTOL-MYERS SQUIBB COMPANY (US) 1993-10-26 US disclosed