SCHEMBL7750652

SCHEMBL7750652

O=C1NC(c2ccc(Cl)c(Cl)c2)=C2C(=O)NC(c3ccc(Cl)cc3)=C12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 4/20 0.43
GSK3B P49841 8/20 0.42
GSK3A P49840 1/20 0.42
MEN1 O00255 2/20 0.42
HTT P42858 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 2/20 0.42
MAPT P10636 2/20 0.42
USP2 O75604 1/20 0.42
PKM P14618 1/20 0.42
ALOX12 P18054 1/20 0.42
PTGS2 P35354 1/20 0.41
TP53 P04637 1/20 0.39
CYP1B1 Q16678 1/20 0.38
NOTUM Q6P988 1/20 0.38
TDP2 O95551 1/20 0.37
CNR1 P21554 1/20 0.37
ALDH1A1 P00352 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286464 0.93 AHR (0.50) AHRGSK3BGSK3AMEN1HTT
SCHEMBL7754317 0.88 AHR (0.42) AHRGSK3BMEN1HTTKMT2A
SCHEMBL91966 0.87 PTGS2 (0.50) GSK3BGSK3AKDM4EGAAMAPT
SCHEMBL12577702 0.87 AHR (0.41) AHRGSK3BGSK3AMEN1HTT
SCHEMBL12424888 0.82 TDP2 (0.51) PTGS2TDP2
SCHEMBL3823878 0.82 PTGS2 (0.56) AHRGSK3BGSK3AMEN1HTT
SCHEMBL13204641 0.81 GSK3B (0.52) GSK3BGSK3ATDP2
SCHEMBL1557806 0.80 GSK3B (0.54) GSK3BMEN1KMT2AKDM4EGAA
SCHEMBL7753950 0.79 CYP2D6 (0.46) GSK3BGSK3AMEN1KMT2AMAPT
SCHEMBL21419776 0.79 GSK3B (0.58) GSK3BGSK3AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765919-B1 Monophasic solid solutions with asymmetrical pyrrolo-(4-3-c)-pyrroles as host CIBA SC HOLDING AG (CH) 2001-02-21 EP disclosed
US-5756746-A KETOPYRROLES AND QUINACRIDONES FOR LIGHT STABLE AND WEATHER RESISTANT COLOR COMPOSITIONS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-05-26 US disclosed
EP-0765919-A2 Monophasic solid solutions with asymmetrical pyrrolo-(4-3-c)-pyrroles as host Ciba SC Holding AG (CH) 1997-04-02 EP disclosed