SCHEMBL7752971

SCHEMBL7752971

CCOP(=O)(Cc1ccc(NC(=O)c2ccc3ccccc3c2)cc1)OCC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.62
MEN1 O00255 4/20 0.62
NR1H4 Q96RI1 2/20 0.60
NPC1 O15118 11/20 0.60
RAB9A P51151 11/20 0.60
CASP3 P42574 3/20 0.60
SENP7 Q9BQF6 3/20 0.60
POLB P06746 1/20 0.57
SENP8 Q96LD8 1/20 0.57
SENP6 Q9GZR1 1/20 0.57
DEGS1 O15121 1/20 0.56
NQO2 P16083 1/20 0.53
KDM4E B2RXH2 1/20 0.52
PLAU P00749 3/20 0.52
F2 P00734 1/20 0.52
PLG P00747 1/20 0.52
PLAT P00750 1/20 0.52
KLKB1 P03952 1/20 0.52
PRSS1 P07477 1/20 0.52
ENPP3 O14638 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537002 0.85 TRPV1 (0.58) KMT2AMEN1NR1H4NPC1RAB9A
SCHEMBL15668082 0.83 PGR (0.60) KMT2AMEN1NR1H4NPC1RAB9A
SCHEMBL9500132 0.81 NPC1 (0.65) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL9499648 0.81 NPC1 (0.59) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL7164864 0.80 NPC1 (0.52) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL9502356 0.80 MAPT (0.55) KMT2AMEN1NPC1KDM4E
SCHEMBL9500932 0.80 RAB9A (0.58) KMT2AMEN1NPC1RAB9ACASP3
SCHEMBL9502383 0.80 HDAC1 (0.50) NPC1RAB9APOLBKDM4E
SCHEMBL10331192 0.79 CYP1A2 (0.52) NPC1RAB9ACASP3SENP7POLB
SCHEMBL7781982 0.79 RAB9A (0.72) KMT2AMEN1NR1H4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0769015-B1 PHOSPHONIC ACID COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-03-14 EP disclosed
US-5716944-A USEFUL AS PROPHYLACTIC AND THERAPEUTIC AGENTS OF VARIOUS METABOLIC BONE DISEASES SUCH AS OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0769015-A1 PHOSPHONIC ACID COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-04-23 EP disclosed
WO-1996001267-A1 PHOSPHONIC ACID COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-01-18 WO disclosed