SCHEMBL7754290

SCHEMBL7754290

O=C1NC(c2ccc(-c3ccccc3)cc2)=C2C(=O)NC(c3ccccc3)=C12

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.48
GSK3B P49841 4/20 0.46
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42
TDP2 O95551 1/20 0.42
ALDH1A1 P00352 1/20 0.41
STK10 O94804 1/20 0.40
SLK Q9H2G2 1/20 0.40
TYRO3 Q06418 1/20 0.39
NTRK2 Q16620 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
CTRC Q99895 1/20 0.39
NAT1 P18440 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91967 1.00 PTGS2 (0.48) PTGS2GSK3BMAOAMAOBSIRT2
SCHEMBL278635 0.95 GSK3B (0.48) PTGS2GSK3BMAOAMAOBALDH1A1
SCHEMBL12577696 0.90 ALDH1A1 (0.56) PTGS2GSK3BMAOAMAOBSIRT2
SCHEMBL92072 0.90 CYP1A2 (0.56) PTGS2GSK3BTDP2CTRC
SCHEMBL12640639 0.90 PTGS2 (0.42) PTGS2GSK3BMAOAMAOBSIRT2
SCHEMBL9833136 0.88 PTGS2 (0.47) PTGS2GSK3BMAOAMAOBALDH1A1
SCHEMBL8502944 0.88 PTGS1 (0.46) PTGS2GSK3BSTK10SLK
SCHEMBL12577691 0.88 ALDH1A1 (0.52) PTGS2GSK3BTDP2ALDH1A1
SCHEMBL1557806 0.88 GSK3B (0.54) PTGS2GSK3B
SCHEMBL13578991 0.86 TAAR1 (0.60) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765919-B1 Monophasic solid solutions with asymmetrical pyrrolo-(4-3-c)-pyrroles as host CIBA SC HOLDING AG (CH) 2001-02-21 EP disclosed
US-5821373-A WITH DIFFERENT 1,4-DIKETOPYRROLOPYRROLE OR QUINACRIDONE; PIGMENTING HIGH MOLECULAR WEIGHT MATERIALS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-10-13 US disclosed
US-5756746-A KETOPYRROLES AND QUINACRIDONES FOR LIGHT STABLE AND WEATHER RESISTANT COLOR COMPOSITIONS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-05-26 US disclosed
EP-0765919-A2 Monophasic solid solutions with asymmetrical pyrrolo-(4-3-c)-pyrroles as host Ciba SC Holding AG (CH) 1997-04-02 EP disclosed