SCHEMBL7754580

SCHEMBL7754580

CC1(C)CCC(C)(C)c2cc(C34CC/C(=C/Cc5ccc(C(=O)O)cn5)C3C4)ccc21

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RXRA P19793 15/20 0.46
RXRB P28702 10/20 0.46
RXRG P48443 8/20 0.46
CYP26A1 O43174 6/20 0.44
CYP26B1 Q9NR63 5/20 0.44
RARB P10826 5/20 0.42
RARG P13631 5/20 0.42
RARA P10276 4/20 0.42
CYP3A4 P08684 2/20 0.42
CRABP2 P29373 1/20 0.42
PPARG P37231 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7754583 1.00 RXRA (0.46) RXRARXRBRXRGCYP26A1CYP26B1
SCHEMBL7756256 0.94 RXRA (0.46) RXRARXRBRXRGCYP26A1CYP26B1
SCHEMBL7756251 0.94 RXRA (0.46) RXRARXRBRXRGCYP26A1CYP26B1
SCHEMBL7756267 0.91 RXRA (0.43) RXRARXRBRXRGCYP26A1CYP26B1
SCHEMBL7756261 0.91 RXRA (0.43) RXRARXRBRXRGCYP26A1CYP26B1
SCHEMBL7789372 0.87 RXRA (0.51) RXRARXRBRXRGRARBRARG
SCHEMBL7789369 0.87 RXRA (0.51) RXRARXRBRXRGRARBRARG
SCHEMBL7756259 0.86 RXRA (0.37) RXRARXRBRXRGCYP26A1CYP26B1
SCHEMBL7757722 0.86 RXRA (0.51) RXRARXRBRXRGCYP26A1CYP26B1
SCHEMBL7757729 0.86 RXRA (0.51) RXRARXRBRXRGCYP26A1CYP26B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20010037025-A1 New compounds, their preparation and use MURRAY ANTHONY (DK) 2001-11-01 US claimed
EP-1077919-A1 NEW COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2001-02-28 EP claimed
WO-1999058486-A1 NEW COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1999-11-18 WO claimed
US-20010037025-A1 New compounds, their preparation and use MURRAY ANTHONY (DK) 2001-11-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010037025-A1 New compounds, their preparation and use GPR119, SLC5A1, SLC5A2 RXRA 874/4885RXRB 1018/4885RXRG 1046/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.