SCHEMBL7754759

SCHEMBL7754759

Cc1c(C(F)(F)F)cnn(-c2cc(F)c(C#N)cc2F)c1=O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.35
PDE2A O00408 2/20 0.34
AR P10275 9/20 0.33
BCAT2 O15382 3/20 0.33
BCAT1 P54687 3/20 0.33
LRRK2 Q5S007 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7754452 0.90 AR (0.33) PDE2AARBCAT2BCAT1
SCHEMBL7753791 0.88 AR (0.38) ARBCAT2BCAT1LRRK2
SCHEMBL7749728 0.86 BCAT2 (0.37) ARBCAT2BCAT1CYP11B1CYP11B2
SCHEMBL7753787 0.83 BCAT2 (0.35) ARBCAT2BCAT1LRRK2
SCHEMBL7753846 0.82 BRD4 (0.35) PDE2AAR
SCHEMBL7755922 0.79 GLA (0.46) ARBCAT2BCAT1KDM4EALDH1A1
SCHEMBL5841567 0.77 RAB9A (0.42) TRPV4BCAT2BCAT1KDM4EALDH1A1
SCHEMBL7754472 0.77 BCL2A1 (0.31) AR
SCHEMBL8570147 0.77 GAA (0.33) GAA
SCHEMBL7753821 0.76 CYP11B1 (0.41) TRPV4ARBCAT2BCAT1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070055-A1 SUBSTITUTED PHENYL PYRIDAZINONES Bayer Aktiengesellschaft (DE) 2001-01-24 EP disclosed
WO-1999052878-A1 SUBSTITUTED PHENYL PYRIDAZINONES BAYER AKTIENGESELLSCHAFT (DE) 1999-10-21 WO disclosed