SCHEMBL7754982

SCHEMBL7754982

CCOC(=O)c1c(O)c2c(OC)c(C)ccc2[nH]c1=O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.52
KDM5B Q9UGL1 1/20 0.52
MAP3K5 Q99683 1/20 0.47
LMNA P02545 1/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 2/20 0.47
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
KDM4E B2RXH2 1/20 0.46
APLNR P35414 1/20 0.46
CSF1R P07333 1/20 0.42
GAA P10253 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL322275 0.88 USP2 (0.44) KDM5AKDM5BALDH1A1MEN1KMT2A
SCHEMBL7828505 0.86 KDM5A (0.48) KDM5AKDM5BMAP3K5LMNAALDH1A1
SCHEMBL321963 0.85 KDM5A (0.54) KDM5AKDM5BMAP3K5LMNAALDH1A1
SCHEMBL7826753 0.84 KDM4E (0.38) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL7754979 0.84 KDM5A (0.53) KDM5AKDM5BMAP3K5LMNAALDH1A1
SCHEMBL1033018 0.84 KDM5A (0.53) KDM5AKDM5BMAP3K5LMNAALDH1A1
SCHEMBL7861387 0.81 KDM5A (0.50) KDM5AKDM5BMAP3K5LMNAALDH1A1
SCHEMBL321856 0.79 KDM5A (0.44) KDM5AKDM5BMAP3K5LMNAALDH1A1
SCHEMBL7556725 0.78 KMT2A (0.43) KDM5AALDH1A1MEN1KMT2AMAPT
SCHEMBL16029767 0.76 MAP3K5 (0.60) KDM5AKDM5BMAP3K5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095021-A1 QUINOLINE DERIVATIVES Active Biotech AB (SE) 2001-05-02 EP disclosed
EP-1073639-A1 QUINOLINE DERIVATIVES Active Biotech AB (SE) 2001-02-07 EP disclosed
WO-2000003991-A1 QUINOLINE DERIVATIVES ACTIVE BIOTECH AB (SE) 2000-01-27 WO disclosed
WO-1999055678-A1 QUINOLINE DERIVATIVES ACTIVE BIOTECH AB (SE) 1999-11-04 WO disclosed