SCHEMBL7756833

SCHEMBL7756833

ClC(Cl)(Cl)c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
CYP2A6 P11509 1/20 0.50
CA2 P00918 4/20 0.39
CA1 P00915 3/20 0.39
CA5A P35218 1/20 0.39
CA9 Q16790 1/20 0.39
ALDH1A1 P00352 4/20 0.38
ALOX15 P16050 2/20 0.38
MAPK1 P28482 2/20 0.38
TDP1 Q9NUW8 1/20 0.35
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
OGG1 O15527 1/20 0.32
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9816151 0.83 TSHR (0.67) TSHRMAPK1TDP1CYP19A1
SCHEMBL545084 0.83 TSHR (0.67) TSHRMAPK1TDP1CYP19A1
SCHEMBL4460794 0.81 CYP2A6 (0.50) TSHRCYP2A6CA2CA1CA5A
SCHEMBL11231213 0.78 TSHR (0.53) TSHRMAPK1
SCHEMBL18548321 0.77 CYP2A6 (0.44) CYP2A6CA2CA1CA5ACA9
SCHEMBL9622508 0.77 CYP2A6 (0.44) TSHRCYP2A6CA2CA1CA5A
SCHEMBL9876029 0.77 CA1 (0.46) TSHRCYP2A6CA2CA1CA5A
SCHEMBL21791779 0.75 CA1 (0.50) TSHRCYP2A6CA2CA1CA5A
SCHEMBL440244 0.73 CYP2A6 (0.57) TSHRCYP2A6CA2CA1CA5A
SCHEMBL28912876 0.73 CYP2A6 (0.57) TSHRCYP2A6CA2CA1CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4163753-A FROM AN ALIPHATIC ACID ANHYDRIDE AND A TRICHLOROMETHYL AROMATIC COMPOUND Diaz Chemical Corporation (US) 1979-08-07 US claimed
US-6313337-B1 Method of making benzoyl halides and nitriles OCCIDENTAL CHEMICAL CORPORATION 2001-11-06 US disclosed
WO-2001079148-A2 METHOD OF MAKING BENZOYL HALIDES AND NITRILES AMERICAN WRECKING CORPORATION OF NEW JERSEY (US) 2001-10-25 WO disclosed
US-4783562-A Process for the preparation of trichloromethyl-substituted aromatic compounds, and trichloromethyl-substituted aromatic compounds obtained in this process BAYER AKTIENGESELLSCHAFT (DE) 1988-11-08 US disclosed
EP-0061029-B1 PROCESS FOR THE PREPARATION OF TRICHLOROMETHYL-SUBSTITUTED AROMATIC COMPOUNDS BAYER AG (DE) 1986-01-08 EP disclosed
EP-0031436-B1 A METHOD FOR THE CLEAVAGE OF SILOXANES HÜLS TROISDORF AKTIENGESELLSCHAFT (DE) 1984-02-15 EP disclosed
US-4383116-A Process for producing 4-benzoylpyrazoles ISHIHARA SANGYO KAISHA LTD. (JP) 1983-05-10 US disclosed
EP-0061029-A1 Process for the preparation of trichloromethyl-substituted aromatic compounds BAYER AG (DE) 1982-09-29 EP disclosed
US-4310680-A METAL OR METAL COMPOUND CATALYST DYNAMIT NOBEL AG (DE) 1982-01-12 US disclosed
EP-0031436-A2 A method for the cleavage of siloxanes HÜLS TROISDORF AKTIENGESELLSCHAFT (DE) 1981-07-08 EP disclosed
US-4220765-A Process for the preparation of 4,6-dihalogeno-triazines BAYER AKTIENGESELLSCHAFT (DE) 1980-09-02 US disclosed
EP-0002493-B1 PROCESS FOR THE PREPARATION OF 4,6-DIHALOGENO-1,3,5-TRIAZINES BAYER AG (DE) 1980-07-23 EP disclosed
US-4163753-A FROM AN ALIPHATIC ACID ANHYDRIDE AND A TRICHLOROMETHYL AROMATIC COMPOUND Diaz Chemical Corporation (US) 1979-08-07 US disclosed