SCHEMBL9876029

SCHEMBL9876029

FC(F)(Cl)c1ccc(Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA5A P35218 1/20 0.46
CA9 Q16790 1/20 0.46
CYP2A6 P11509 1/20 0.44
TRPV1 Q8NER1 1/20 0.35
ALDH1A1 P00352 4/20 0.35
ALOX15 P16050 2/20 0.35
MAPK1 P28482 2/20 0.35
AHR P35869 2/20 0.33
TDP1 Q9NUW8 1/20 0.32
GSK3B P49841 1/20 0.31
TSHR P16473 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
NT5E P21589 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4204801 0.85 PDE2A (0.36) ALDH1A1MAPK1AHRGSK3BTSHR
Hydrochloric Acid SCHEMBL8577339 0.82 PDE2A (0.35) ALDH1A1MAPK1AHRGSK3BTSHR
Hydrochloric Acid SCHEMBL8577343 0.82 PDE2A (0.35) ALDH1A1MAPK1AHRGSK3BTSHR
SCHEMBL7756833 0.77 TSHR (0.50) CA1CA2CA5ACA9CYP2A6
SCHEMBL21791779 0.77 CA1 (0.50) CA1CA2CA5ACA9CYP2A6
SCHEMBL1508480 0.77 ALDH1A1 (0.50) ALDH1A1AHRGSK3BTSHRCES2
SCHEMBL4460794 0.77 CYP2A6 (0.50) CA1CA2CA5ACA9CYP2A6
SCHEMBL11240836 0.77 PDE2A (0.32) ALDH1A1MAPK1TSHR
SCHEMBL8909 0.77 TRPV1 (0.50) CA1CA2CA5ACA9CYP2A6
SCHEMBL3675742 0.77 CA1 (0.50) CA1CA2CA5ACA9CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990657-A From an aromatic halide without a phase transfer agent RHONE-POULENC CHIMIE (FR) 1991-02-05 US disclosed
EP-0255794-A1 Process for preparing an aromatic acid RHONE-POULENC CHIMIE (FR) 1988-02-10 EP disclosed
EP-0109606-B1 PROCESS FOR THE FORMYLATION OF ARYL HALIDES BAYER AG (DE) 1986-01-22 EP disclosed
US-4536344-A USING A PHOSPINE OR PHOSPHITE BAYER AKTIENGESELLSCHAFT (DE) 1985-08-20 US disclosed
EP-0109606-A1 Process for the formylation of aryl halides BAYER AG (DE) 1984-05-30 EP disclosed