SCHEMBL7756903

SCHEMBL7756903

COc1ccc(COc2ccccc2NC(=O)NCCN)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.53
HDAC1 Q13547 2/20 0.52
HDAC3 O15379 1/20 0.52
HDAC2 Q92769 1/20 0.52
NCOR2 Q9Y618 1/20 0.52
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MAPK1 P28482 1/20 0.51
BLM P54132 1/20 0.51
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
MAPT P10636 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
GAA P10253 1/20 0.50
FPR2 P25090 1/20 0.50
HDAC6 Q9UBN7 1/20 0.49
USP2 O75604 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7756925 0.86 NPC1 (0.49) BRD4HDAC1HDAC3HDAC2NCOR2
SCHEMBL8366817 0.84 BRD4 (0.59) BRD4HDAC1HDAC3HDAC2NCOR2
SCHEMBL7760029 0.82 NPC1 (0.67) BRD4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL7756878 0.81 KDM4E (0.58) HDAC1HDAC3HDAC2NCOR2NPC1
SCHEMBL7760871 0.81 PLA2G1B (0.57) BRD4NPC1RAB9ASMN1; SMN2MAPK1
SCHEMBL7760879 0.78 MAPT (0.53) HDAC1HDAC3HDAC2NPC1RAB9A
Hydrochloric Acid SCHEMBL6771484 0.74 HDAC3 (0.55) BRD4HDAC1HDAC3HDAC2NCOR2
SCHEMBL3585982 0.74 HDAC8 (0.55) BRD4HDAC1HDAC3HDAC2RAB9A
SCHEMBL13366908 0.73 CASR (0.63) HDAC1NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL321103 0.73 LTA4H (0.68) NPC1RAB9ASMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6541479-B1 Derivatives of thiosalicylic acid and o-aminobenzoic acid MASSACHUSETTS COLLEGE OF PHARMACY 2003-04-01 US disclosed