SCHEMBL7761017

SCHEMBL7761017

CC(=O)O[C@@H](CCCNCc1ccccc1)[C@@H](C)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
NCOR2 Q9Y618 2/20 0.43
MAOA P21397 1/20 0.43
CHRM2 P08172 1/20 0.42
KDM4E B2RXH2 2/20 0.41
MITF O75030 1/20 0.41
GAA P10253 1/20 0.41
FOLH1 Q04609 1/20 0.41
CTSK P43235 3/20 0.41
CTSL P07711 2/20 0.41
CTSB P07858 2/20 0.41
CTSH P09668 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CCR6 P51684 1/20 0.41
PAX8 Q06710 1/20 0.41
MAPK1 P28482 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7761961 1.00 HDAC3 (0.43) HDAC3HDAC1HDAC2HDAC8NCOR2
Trifluoroacetic Acid SCHEMBL9080870 0.94 KDM4E (0.42) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL7763332 0.83 TRPA1 (0.42) CTSKCTSLCTSBCTSHALDH1A1
SCHEMBL7763374 0.83 TRPA1 (0.46) CTSKCTSLCTSBCTSHALDH1A1
SCHEMBL7760075 0.83 TRPA1 (0.46) CTSKCTSLCTSBCTSHALDH1A1
SCHEMBL7760073 0.83 TRPA1 (0.42) CTSKCTSLCTSBCTSHALDH1A1
SCHEMBL12358871 0.82 CTSK (0.42) CTSKCTSLCTSBCTSHMEN1
SCHEMBL7779594 0.80 TRPA1 (0.46) HDAC3HDAC1HDAC2HDAC8CTSK
SCHEMBL7756946 0.79 TRPA1 (0.44) ALDH1A1
SCHEMBL12358872 0.78 FDFT1 (0.41) CTSKCTSLCTSBCTSH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821665-B1 CYCLOBUTANE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHASE AND PROTEIN FARNESYLTRANSFERASE ABBOTT LAB (US) 2001-10-04 EP disclosed
EP-1090908-A2 Cyclobutane derivatives as inhibitors of protein farnesyltransferase ABBOTT LABORATORIES (US) 2001-04-11 EP disclosed