SCHEMBL7760073

SCHEMBL7760073

CC(=O)O[C@@H](CCCI)[C@@H](C)Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.42
FDFT1 P37268 3/20 0.41
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CTSK P43235 3/20 0.39
CTSL P07711 2/20 0.39
CTSB P07858 2/20 0.39
CTSH P09668 2/20 0.39
ALDH1A1 P00352 1/20 0.39
ALPI P09923 1/20 0.39
PKM P14618 1/20 0.39
PTGS1 P23219 1/20 0.39
XIAP P98170 1/20 0.39
SLC7A5 Q01650 1/20 0.39
LMNA P02545 1/20 0.38
TRPV1 Q8NER1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7763332 1.00 TRPA1 (0.42) TRPA1FDFT1CYP2D6TSHRNPC1
SCHEMBL7763374 0.89 TRPA1 (0.46) TRPA1FDFT1CYP2D6TSHRNPC1
SCHEMBL7760075 0.89 TRPA1 (0.46) TRPA1FDFT1CYP2D6TSHRNPC1
SCHEMBL7779594 0.85 TRPA1 (0.46) TRPA1FDFT1CYP2D6TSHRNPC1
SCHEMBL12358871 0.85 CTSK (0.42) TRPA1FDFT1CYP2D6TSHRNPC1
SCHEMBL7756946 0.84 TRPA1 (0.44) TRPA1FDFT1CYP2D6TSHRNPC1
SCHEMBL7761961 0.83 HDAC3 (0.43) CTSKCTSLCTSBCTSHALDH1A1
SCHEMBL7761017 0.83 HDAC3 (0.43) CTSKCTSLCTSBCTSHALDH1A1
SCHEMBL12358872 0.81 FDFT1 (0.41) TRPA1FDFT1CTSKCTSLCTSB
SCHEMBL2600696 0.81 TRPA1 (0.46) TRPA1FDFT1CYP2D6TSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821665-B1 CYCLOBUTANE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHASE AND PROTEIN FARNESYLTRANSFERASE ABBOTT LAB (US) 2001-10-04 EP disclosed
EP-1090908-A2 Cyclobutane derivatives as inhibitors of protein farnesyltransferase ABBOTT LABORATORIES (US) 2001-04-11 EP disclosed
US-5831115-A CYCLOBUTANECARBOXAMIDES ABBOTT LABORATORIES (US) 1998-11-03 US disclosed