SCHEMBL7764412

SCHEMBL7764412

c1cc(NC2CCCCC2)ncn1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.55
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
CTSK P43235 1/20 0.51
MALT1 Q9UDY8 1/20 0.51
GAA P10253 1/20 0.48
HCAR3 P49019 2/20 0.46
MKNK1 Q9BUB5 1/20 0.46
AURKB Q96GD4 1/20 0.43
EPHX1 P07099 1/20 0.42
AOC1 P19801 2/20 0.42
AOC3 Q16853 2/20 0.42
SCN9A Q15858 1/20 0.42
MAP4K4 O95819 1/20 0.42
S1PR3 Q99500 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29779677 0.98 S1PR1 (0.52) S1PR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL23304369 0.94 MALT1 (0.52) S1PR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL1671847 0.90 MALT1 (0.58) S1PR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL14520680 0.82 MALT1 (0.52) S1PR1MEN1KMT2AALDH1A1MALT1
SCHEMBL29501368 0.82 HRH3 (0.58) S1PR1MEN1KMT2AALDH1A1MALT1
SCHEMBL25426946 0.82 MAPK1 (0.51) S1PR1MEN1KMT2AALDH1A1MALT1
SCHEMBL4006284 0.82 HRH3 (0.58) S1PR1MEN1KMT2AALDH1A1MALT1
SCHEMBL2051027 0.80 PRKCZ (0.50)
SCHEMBL14980406 0.80 MALT1 (0.50) KDM4EALDH1A1L3MBTL1MALT1
SCHEMBL31127364 0.80 MALT1 (0.47) S1PR1MALT1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022059996-A1 BLOOD CIRCULATION MICRO IN-VITRO CORPUSCLE-MEDIATED CANCER TREATMENT COMPOSITION 서울대학교 기술지주 주식회사 2022-03-24 WO disclosed
EP-3405466-B1 ARYL SUBSTITUTED PYRIMIDINES FOR USE IN INFLUENZA VIRUS INFECTION JANSSEN SCIENCES IRELAND UNLIMITED CO (IE) 2020-11-18 EP disclosed
WO-2017125506-A1 ARYL SUBSTITUTED PYRIMIDINES FOR USE IN INFLUENZA VIRUS INFECTION JANSSEN SCIENCES IRELAND UC (IE) 2017-07-27 WO disclosed
EP-1100785-A1 SUBSTITUTED CYCLOHEXYLAMINOPYRIMIDINES Aventis CropScience GmbH (DE) 2001-05-23 EP disclosed
US-6197729-B1 COMBATING PEST WHICH COMPRISES APPLYING TO PEST OR ITS LOCUS PESTICIDAL CYCLOHEXYLAMINOPYRIMIDINNE COMPOUND HOECHST SCHERING AGREVO (DE) 2001-03-06 US disclosed
WO-2000007998-A1 SUBSTITUTED CYCLOHEXYLAMINOPYRIMIDINES AVENTIS CROPSCIENCE GMBH (DE) 2000-02-17 WO disclosed
WO-1996006086-A1 4-CYCLOHEXYLAMINOPYRIMIDINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND AGROHORTICULTURAL PEST CONTROL DRUG UBE INDUSTRIES, LTD. (JP) 1996-02-29 WO disclosed