SCHEMBL7765708

SCHEMBL7765708

COc1ccc2c(c1)C(CO)=Cc1ccccc1O2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.41
LMNA P02545 2/20 0.39
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
CYP19A1 P11511 1/20 0.37
HDAC3 O15379 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
HDAC4 P56524 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
HDAC1 Q13547 1/20 0.37
TUBB2A Q13885 1/20 0.37
TUBB8 Q3ZCM7 1/20 0.37
TUBA3E Q6PEY2 1/20 0.37
TUBA1A Q71U36 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7769544 0.86 TRPA1 (0.41) TRPA1LMNAHTR2AHTR2CCYP19A1
SCHEMBL5952981 0.84 TRPA1 (0.39) TRPA1LMNAHTR2AHTR2CCYP19A1
SCHEMBL5953534 0.84 HTR2A (0.44) TRPA1LMNAHTR2AHTR2CCYP19A1
SCHEMBL6685325 0.79 DRD2 (0.44) TRPA1LMNAMAPTTDP1KDM4E
SCHEMBL5953348 0.78 DRD2 (0.48) MAPTTDP1KDM4EDRD2DRD4
SCHEMBL7770756 0.78 LMNA (0.60) TRPA1LMNACYP19A1HDAC3TUBB4A
SCHEMBL5953775 0.78 PYCR1 (0.45) TRPA1LMNAHTR2AHTR2CSMN1; SMN2
SCHEMBL9630555 0.76 MEN1 (0.42) MAPTSMN1; SMN2KDM4ENPC1ALDH1A1
SCHEMBL7770761 0.75 LMNA (0.44) TRPA1LMNACYP19A1HDAC3TUBB4A
Metoxepin SCHEMBL2109740 0.72 DRD2 (0.70) HTR2AHTR2CMAPTTDP1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726265-B1 10-Aminoaliphatyl-dibenz(b,f)oxepins with antineurodegenarative activity NOVARTIS AG (CH) 2001-07-25 EP disclosed
EP-0726265-A1 10-Aminoaliphatyl-dibenz(b,f)oxepins with antineurodegenarative activity CIBA-GEIGY AG (CH) 1996-08-14 EP disclosed