SCHEMBL7765918

SCHEMBL7765918

COC(=O)NC(=O)[C@@H](N)CCSC

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.39
METAP1 P53582 1/20 0.39
SLC15A1 P46059 1/20 0.39
CTSC P53634 2/20 0.38
RNPEP Q9H4A4 1/20 0.36
MARS1 P56192 5/20 0.36
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
ANPEP P15144 1/20 0.34
ENPEP Q07075 1/20 0.34
FNTA P49354 3/20 0.34
FNTB P49356 3/20 0.34
PGGT1B P53609 1/20 0.34
ARG1 P05089 1/20 0.34
ARG2 P78540 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7766597 1.00 METAP2 (0.39) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL17746783 0.87 SLC15A1 (0.48) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL7766540 0.86 METAP2 (0.50) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL7762932 0.86 METAP2 (0.50) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL538813 0.81 SLC15A1 (0.41) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL11032201 0.81 ALDH1A1 (0.41) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL2342221 0.81 ALDH1A1 (0.41) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL538814 0.81 SLC15A1 (0.41) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL2342224 0.81 ALDH1A1 (0.41) METAP2METAP1SLC15A1CTSCRNPEP
SCHEMBL23692301 0.77 RNPEP (0.39) METAP2METAP1SLC15A1CTSCRNPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759066-A1 PROCESS FOR OBTAINING MICRO-ORGANISMS CONTAINING PEPTIDE AMIDASE, MICRO-ORGANISMS OBTAINED THEREWITH, PEPTIDE AMIDASES CONTAINED IN THEM AND USE THEREOF Degussa Aktiengesellschaft (DE) 1997-02-26 EP claimed
WO-1995030740-A1 PROCESS FOR OBTAINING MICRO-ORGANISMS CONTAINING PEPTIDE AMIDASE, MICRO-ORGANISMS OBTAINED THEREWITH, PEPTIDE AMIDASES CONTAINED IN THEM AND USE THEREOF DEGUSSA AKTIENGESELLSCHAFT (DE) 1995-11-16 WO claimed
EP-0759066-B1 PROCESS FOR OBTAINING MICRO-ORGANISMS CONTAINING PEPTIDE AMIDASE, MICRO-ORGANISMS OBTAINED THEREWITH, PEPTIDE AMIDASES CONTAINED IN THEM AND USE THEREOF DEGUSSA (DE) 2001-06-27 EP disclosed
EP-0759066-A1 PROCESS FOR OBTAINING MICRO-ORGANISMS CONTAINING PEPTIDE AMIDASE, MICRO-ORGANISMS OBTAINED THEREWITH, PEPTIDE AMIDASES CONTAINED IN THEM AND USE THEREOF Degussa Aktiengesellschaft (DE) 1997-02-26 EP disclosed
WO-1995030740-A1 PROCESS FOR OBTAINING MICRO-ORGANISMS CONTAINING PEPTIDE AMIDASE, MICRO-ORGANISMS OBTAINED THEREWITH, PEPTIDE AMIDASES CONTAINED IN THEM AND USE THEREOF DEGUSSA AKTIENGESELLSCHAFT (DE) 1995-11-16 WO disclosed