SCHEMBL7768288

SCHEMBL7768288

Oc1cccc2sc(-c3ccc(OCCN4CCCC4)cc3)cc12

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.56
ESR1 P03372 13/20 0.56
ESR2 Q92731 13/20 0.56
LTA4H P09960 2/20 0.53
CHEK1 O14757 1/20 0.51
F2 P00734 1/20 0.51
HRH3 Q9Y5N1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7768257 0.84 ESR1 (0.56) ITGA4ESR1ESR2LTA4HCHEK1
SCHEMBL6594650 0.82 LTA4H (0.60) ITGA4LTA4HHRH3
SCHEMBL7441443 0.81 ESR1 (0.56) ESR1ESR2LTA4HCHEK1HRH3
SCHEMBL7773130 0.78 ESR1 (0.55) ESR1ESR2CHEK1F2
SCHEMBL7451900 0.75 ESR1 (0.84) ITGA4ESR1ESR2F2
SCHEMBL6595152 0.74 LTA4H (0.55) ESR1ESR2LTA4HHRH3
SCHEMBL6593929 0.74 ESR1 (0.56) ESR1ESR2LTA4HHRH3
SCHEMBL7774143 0.74 LTA4H (0.55) ITGA4ESR1ESR2LTA4HCHEK1
SCHEMBL6597298 0.74 ACHE (0.54) ESR1ESR2LTA4HCHEK1HRH3
SCHEMBL7436764 0.74 LTA4H (0.71) ESR1ESR2LTA4HHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed