SCHEMBL7775378

SCHEMBL7775378

Cc1cnc(N2C[CH]NCC2)nc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GPR119 Q8TDV5 2/20 0.35
TAAR1 Q96RJ0 1/20 0.34
DHFR P00374 1/20 0.34
OGA O60502 1/20 0.34
KCNH2 Q12809 1/20 0.33
BPTF Q12830 1/20 0.33
HTR1A P08908 2/20 0.33
HTR1D P28221 2/20 0.33
HTR1B P28222 2/20 0.33
HTR7 P34969 2/20 0.33
HTR2B P41595 2/20 0.33
HTR6 P50406 2/20 0.33
HTR5A P47898 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356574 0.79 ALDH1A1 (0.57) ALDH1A1KDM4ECYP1A2CYP3A4HPGD
SCHEMBL7991455 0.77 ALDH1A1 (0.59) ALDH1A1KDM4ETAAR1BPTFHTR1A
Hydrochloric Acid SCHEMBL28966659 0.76 ALDH1A1 (0.62) ALDH1A1KDM4ETAAR1BPTFHTR1A
SCHEMBL14161699 0.70 ROCK2 (0.41) GPR119
SCHEMBL23560718 0.70 ROCK2 (0.41) GPR119
SCHEMBL436107 0.70 POLB (0.47) ALDH1A1GPR119DHFROGAKCNH2
SCHEMBL12457554 0.70 GPR119 (0.44) ALDH1A1KDM4EGPR119DHFROGA
SCHEMBL19117494 0.69 AOC3 (0.49) ALDH1A1KDM4EGPR119OGAKCNH2
SCHEMBL10085632 0.69 SMN1; SMN2 (0.50) ALDH1A1GPR119DHFROGAKCNH2
SCHEMBL22538719 0.68 HTR1A (0.41) ALDH1A1KDM4EHTR1AHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117663-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2001-07-25 EP disclosed
WO-2000018767-A9 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORP (US) 2001-04-19 WO disclosed
WO-2000018767-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-04-06 WO disclosed