SCHEMBL7775969

SCHEMBL7775969

COc1cc(C(=O)c2c(N(C)C)sc3ccccc23)ccc1CN1CCOCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.43
KDM4E B2RXH2 5/20 0.42
MAPT P10636 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 2/20 0.42
MAPK1 P28482 2/20 0.42
HTT P42858 2/20 0.42
MITF O75030 1/20 0.42
ALOX15 P16050 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
BCHE P06276 2/20 0.41
ACHE P22303 2/20 0.41
ALDH1A1 P00352 1/20 0.41
RECQL P46063 1/20 0.41
CNR1 P21554 2/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
KCNJ1 P48048 1/20 0.40
CNR2 P34972 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423819 0.92 ESR1 (0.48) KDM4ESMN1; SMN2BCHEACHEALDH1A1
SCHEMBL6171651 0.86 EGFR (0.42) KDM4EMAPTSMN1; SMN2LMNAHTT
SCHEMBL7775991 0.80 ESR1 (0.55) CNR1ESR1ESR2CNR2
SCHEMBL6599641 0.80 ESR1 (0.41) TP53KDM4EMAPTSMN1; SMN2LMNA
SCHEMBL7768296 0.79 ESR1 (0.71) ESR1ESR2
SCHEMBL6171046 0.78 CD274 (0.44) KDM4ETDP1ALDH1A1ESR1ESR2
SCHEMBL6172000 0.76 ESR1 (0.61) TP53MAPTLMNAALOX15TDP1
SCHEMBL6172361 0.75 HTR6 (0.41) CNR1ESR1ESR2CNR2
SCHEMBL221039 0.74 KCNJ1 (0.54) KDM4EMAPTSMN1; SMN2LMNAMAPK1
SCHEMBL1012433 0.74 L3MBTL1 (0.60) TP53KDM4EMAPTSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed