SCHEMBL7778464

SCHEMBL7778464

O=C(O)N1CCCCN1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
ATM Q13315 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HPGD P15428 3/20 0.32
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
GAA P10253 1/20 0.31
CA2 P00918 1/20 0.31
CHKA P35790 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
DPP7 Q9UHL4 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8612756 0.97 ALDH1A1 (0.43) ALDH1A1ATMCYP1A2MAPK1SMN1; SMN2
SCHEMBL3037561 0.93 ALDH1A1 (0.36) ALDH1A1
SCHEMBL29237189 0.76 ALDH1A1 (0.44) ALDH1A1ATMSMN1; SMN2HPGDMMP1
SCHEMBL7779646 0.76 TSHR (0.41) ALDH1A1ATMSMN1; SMN2GAAPOLB
SCHEMBL4106642 0.74 CTSK (0.50)
SCHEMBL28449030 0.74
SCHEMBL76824 0.71
Bromide SCHEMBL1732225 0.69
SCHEMBL6704420 0.69 ALDH1A1 (0.58) ALDH1A1ATMHPGDMMP1MMP2
SCHEMBL336899 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0693482-B1 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE AND HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLATE DERIVATIVE IHARA CHEMICAL IND CO (JP) 2001-09-12 EP disclosed
EP-0693482-B1 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE AND HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLATE DERIVATIVE IHARA CHEMICAL IND CO (JP) 2001-09-12 EP disclosed
US-6194577-B1 OXIDIZING 1-AMINOPYRROLIDINE IN PRESENCE OF INORGANIC BASE WITH AIR, OXYGEN OR AQUEOUS HYDROGEN PEROXIDE AS AN OXIDIZING AGENT TO FORM TETRAHYDROPYRIDAZINE JAPAN HYDRAZINE CO., LTD. (JP) 2001-02-27 US disclosed
US-5977360-A Process for producing cyclic hydrazine derivatives, tetra-hydropyridazine and hexahydropyridazine JAPAN HYDRAZINE CO., LTD. (JP) 1999-11-02 US disclosed
US-5872253-A MULTISTAGE PROCESS WITH REACTION OF ISOTHIOCYANATE WITH AMINE AND CYCLIZATION THE THIOUREA WITH HALOCARBONYL HALIDE AMERICAN CYANAMID COMPANY (US) 1999-02-16 US disclosed
EP-0850930-A2 A process for producing alicyclic hydrazine derivatives, tetra-hydropyridazine and hexahydropyridazine JAPAN HYDRAZINE CO., LTD. (JP) 1998-07-01 EP disclosed
US-5726126-A 1-(3-heterocyclyphenyl)-S-triazine-2,6,6-oxo or thiotrione herbicidal agents AMERICAN CYANAMID COMPANY (US) 1998-03-10 US disclosed
US-5705644-A 1-(3-heterocyclphenyl)-s-triazine-2,4,6-oxo or thiotrione herbicidal agents AMERICAN CYANAMID COMPANY (US) 1998-01-06 US disclosed
US-5679791-A FROM A CORRESPONDING ISOTHIOCYANATE COMPOUNDS AND A HYDRAZINE COMPOUND AMERICAN CYANAMID COMPANY (US) 1997-10-21 US disclosed
US-5659031-A CONTROLLING WEEDS IN CROPS AMERICAN CYANAMID COMPANY (US) 1997-08-19 US disclosed
US-5616706-A PREEMERGENCE OR POSTEMERGENCE AMERICAN CYANAMID COMPANY (US) 1997-04-01 US disclosed
US-5612481-A 1-(3-heterocyclylphenyl)-s-triazine-2,4,6-oxo or thiortione herbicidal agents AMERICAN CYANAMID COMPANY (US) 1997-03-18 US disclosed
US-5610120-A APPLYING COMPOUND TO FOLIAGE OF UNDESIRABLE PLANTS OR TO THE SOIL OR WATER CONTAINING SEEDS THEREOF AMERICAN CYANAMID COMPANY (US) 1997-03-11 US disclosed
EP-0745599-A2 1-(3-Heterocyclylphenyl)-s-triazine-2,4,6-oxo or thiotrione herbicidal agents American Cyanamid Company (US) 1996-12-04 EP disclosed
EP-0693482-A4 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE AND HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLATE DERIVATIVE IHARA CHEMICAL IND CO (JP) 1996-04-10 EP disclosed
EP-0693482-A1 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE AND HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLATE DERIVATIVE IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1996-01-24 EP disclosed
EP-0693482-A1 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE AND HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLATE DERIVATIVE IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1996-01-24 EP disclosed
WO-1995021828-A1 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE AND HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLATE DERIVATIVE IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-08-17 WO disclosed
EP-0519083-A1 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLIC ACID DERIVATIVE IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1992-12-23 EP disclosed
WO-1992012136-A1 PROCESS FOR PRODUCING HEXAHYDROPYRIDAZINE-1,2-DICARBOXYLIC ACID DERIVATIVE IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1992-07-23 WO disclosed