SCHEMBL7780080

SCHEMBL7780080

COc1cccc(C(N[C@@H](C)c2cccc(F)c2)c2cccc(N)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
CYP3A4 P08684 1/20 0.46
PFKFB3 Q16875 1/20 0.46
CASR P41180 5/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
AOC3 Q16853 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
LMNA P02545 2/20 0.40
GAA P10253 1/20 0.40
NFE2L2 Q16236 1/20 0.40
POLB P06746 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ROCK2 O75116 1/20 0.38
EGFR P00533 1/20 0.38
KRAS P01116 1/20 0.38
SOS1 Q07889 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7780790 0.91 ALDH1A1 (0.50) ALDH1A1CYP3A4PFKFB3CASRKMT2A
SCHEMBL7785107 0.91 ALDH1A1 (0.50) ALDH1A1CYP3A4PFKFB3CASRKMT2A
SCHEMBL27530316 0.91 ALDH1A1 (0.50) ALDH1A1CYP3A4PFKFB3CASRKMT2A
SCHEMBL7780421 0.87 CASR (0.51) ALDH1A1CYP3A4CASRMEN1KMT2A
SCHEMBL7780426 0.85 SLC6A2 (0.41) ALDH1A1CASRMEN1KMT2ALMNA
SCHEMBL28746788 0.85 SLC6A2 (0.41) ALDH1A1CASRMEN1KMT2ALMNA
SCHEMBL7787788 0.84 CASR (0.37) ALDH1A1CASRLMNAGAA
SCHEMBL7785574 0.84 ALDH1A1 (0.45) ALDH1A1CYP3A4CASRKMT2ALMNA
SCHEMBL7785570 0.84 KMT2A (0.40) ALDH1A1CYP3A4PFKFB3CASRMEN1
SCHEMBL7785129 0.84 ALDH1A1 (0.45) ALDH1A1CYP3A4CASRKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed