SCHEMBL7787788

SCHEMBL7787788

C[C@@H](NC(c1ccc(F)cc1)c1cccc(N)c1)c1cccc(F)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.37
SLC6A9 P48067 1/20 0.37
SLC6A5 Q9Y345 1/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
KCNK3 O14649 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
MAPK1 P28482 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
MTOR P42345 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28746788 0.93 SLC6A2 (0.41) CASRCES2CES1ALDH1A1LMNA
SCHEMBL7780426 0.93 SLC6A2 (0.41) CASRCES2CES1ALDH1A1LMNA
SCHEMBL7785487 0.92 CASR (0.36) CASRCES2CES1ALDH1A1LMNA
SCHEMBL7787615 0.92 MAPKAPK2 (0.33) SLC6A9SLC6A5MAPKAPK2SLC6A2SLC6A4
SCHEMBL7785653 0.91 SLC6A2 (0.36) CASRSLC6A2SLC6A4
SCHEMBL7785680 0.90 NPC1 (0.41) SLC6A9SLC6A5ALDH1A1LMNAGAA
SCHEMBL7785234 0.89 MAPKAPK2 (0.34) SLC6A9SLC6A5ALDH1A1MAPKAPK2SLC6A2
SCHEMBL7780509 0.89 MAPKAPK2 (0.34) SLC6A9SLC6A5ALDH1A1MAPKAPK2SLC6A2
SCHEMBL7780790 0.89 ALDH1A1 (0.50) CASRALDH1A1LMNAGAA
SCHEMBL7785107 0.89 ALDH1A1 (0.50) CASRALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed