SCHEMBL7780426

SCHEMBL7780426

C[C@@H](NC(c1ccccc1)c1cccc(N)c1)c1cccc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
MTOR P42345 1/20 0.40
GPR139 Q6DWJ6 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
CASR P41180 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
MAPKAPK2 P49137 1/20 0.36
CNR2 P34972 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28746788 1.00 SLC6A2 (0.41) SLC6A2SLC6A4IDO1TDO2MTOR
SCHEMBL7787788 0.93 CASR (0.37) SLC6A2SLC6A4IDO1TDO2MTOR
SCHEMBL7780536 0.91 IDO1 (0.39) SLC6A2SLC6A4IDO1TDO2MTOR
SCHEMBL7780766 0.91 IDO1 (0.39) SLC6A2SLC6A4IDO1TDO2MTOR
SCHEMBL7785487 0.91 CASR (0.36) SLC6A2SLC6A4ALDH1A1LMNAGAA
SCHEMBL7785653 0.89 SLC6A2 (0.36) SLC6A2SLC6A4CASRCNR2MEN1
SCHEMBL7785680 0.89 NPC1 (0.41) MTORGPR139ALDH1A1LMNAGAA
SCHEMBL7784931 0.88 SIGMAR1 (0.42) ALDH1A1LMNAGAAMAPKAPK2MEN1
SCHEMBL7780579 0.88 SIGMAR1 (0.42) ALDH1A1LMNAGAAMAPKAPK2MEN1
SCHEMBL7785107 0.87 ALDH1A1 (0.50) ALDH1A1LMNAGAACASRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed