SCHEMBL7780158

SCHEMBL7780158

CC(C)(c1cccc(C(F)(F)F)c1)c1cc(Cl)ncn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.40
KCNQ3 O43525 2/20 0.39
KCNQ2 O43526 2/20 0.39
KCNE1 P15382 2/20 0.39
KCNQ1 P51787 2/20 0.39
KCNQ5 Q9NR82 1/20 0.37
CES2 O00748 1/20 0.37
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK5 Q00535 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDK5R1 Q15078 1/20 0.36
DYRK2 Q92630 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
KDM4E B2RXH2 1/20 0.36
KMO O15229 1/20 0.36
TSHR P16473 2/20 0.36
MAPK1 P28482 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7781185 0.77 BRAF (0.39) THRBCES2TSHRMAPK1CA1
SCHEMBL7775883 0.76 MAPT (0.48) MAPK1ALDH1A1POLB
SCHEMBL1660333 0.74 CA2 (0.39) CA2
SCHEMBL1661082 0.73 CA2 (0.38) CA2
SCHEMBL17663 0.72 CA2 (0.56) KDM4ECA2ALDH1A1
SCHEMBL601224 0.72 KMO (0.61) THRBCCNA2CDK2CDK5DYRK1A
SCHEMBL16532258 0.71 CA2 (0.36) CA2
SCHEMBL7776085 0.70 KDR (0.43)
SCHEMBL7776064 0.70 HTR2B (0.46)
SCHEMBL31750237 0.70 HTR2B (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0972770-B1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof BASF AG (DE) 2001-09-19 EP disclosed
US-6281219-B1 4,6-BIS-ARYL-PYRIMIDINES WHEREIN THE AROMATIC GROUPS ARE ATTACHED VIA TWO LINKING GROUPS WHICH ARE DIFFERENT FROM ONE ANOTHER. AMERICAN CYANAMID CO. 2001-08-28 US disclosed
EP-0972770-A1 Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof American Cyanamid Company (US) 2000-01-19 EP disclosed