SCHEMBL7780321

SCHEMBL7780321

COc1ccc(C(N[C@H](C)c2ccc(F)cc2)c2cccc(N)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.48
ALDH1A1 P00352 5/20 0.48
LMNA P02545 4/20 0.48
HTT P42858 2/20 0.48
MITF O75030 2/20 0.48
MAPT P10636 1/20 0.48
GAA P10253 2/20 0.46
MEN1 O00255 4/20 0.41
ATM Q13315 1/20 0.41
ACP3 P15309 2/20 0.41
SLC6A9 P48067 2/20 0.40
SLC6A5 Q9Y345 2/20 0.40
CYP3A4 P08684 2/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ACHE P22303 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CRHBP P24387 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7784989 0.94 ACP3 (0.45) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL27530316 0.91 ALDH1A1 (0.50) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL7785129 0.91 ALDH1A1 (0.45) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL7785107 0.91 ALDH1A1 (0.50) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL7785570 0.91 KMT2A (0.40) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL7785574 0.91 ALDH1A1 (0.45) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL7780790 0.91 ALDH1A1 (0.50) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL7780316 0.91 ACP3 (0.49) KMT2AALDH1A1LMNAHTTMITF
SCHEMBL7780312 0.89 ACP3 (0.41) KMT2AALDH1A1LMNAMAPTGAA
SCHEMBL7785680 0.88 NPC1 (0.41) KMT2AALDH1A1LMNAHTTMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed