SCHEMBL7785680

SCHEMBL7785680

C[C@@H](NC(c1ccc(F)cc1)c1cccc(N)c1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 2/20 0.39
MITF O75030 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
MTOR P42345 1/20 0.37
EGFR P00533 2/20 0.37
HTR7 P34969 2/20 0.37
GAA P10253 2/20 0.36
GPR139 Q6DWJ6 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
SLC6A9 P48067 1/20 0.36
SLC6A5 Q9Y345 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7784931 0.91 SIGMAR1 (0.42) ALDH1A1KDM4ECYP3A4LMNAMAPT
SCHEMBL7780579 0.91 SIGMAR1 (0.42) ALDH1A1KDM4ECYP3A4LMNAMAPT
SCHEMBL7787615 0.90 MAPKAPK2 (0.33) NPC1CYP3A4CYP2D6SLC6A9SLC6A5
SCHEMBL7787788 0.90 CASR (0.37) ALDH1A1LMNAMTORGAASLC6A9
SCHEMBL7780536 0.89 IDO1 (0.39) ALDH1A1LMNAMTORGAAGPR139
SCHEMBL28746788 0.89 SLC6A2 (0.41) ALDH1A1LMNAKMT2AMTORGAA
SCHEMBL7780766 0.89 IDO1 (0.39) ALDH1A1LMNAMTORGAAGPR139
SCHEMBL7780426 0.89 SLC6A2 (0.41) ALDH1A1LMNAKMT2AMTORGAA
SCHEMBL7780321 0.88 KMT2A (0.48) ALDH1A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7785470 0.88 TRPM8 (0.32) NPC1ALDH1A1CYP3A4CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed