SCHEMBL7780329

SCHEMBL7780329

CCC(NC(c1ccc(OC)cc1)c1cccc(N)c1)c1ccc(F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
CYP3A4 P08684 2/20 0.39
AOC3 Q16853 3/20 0.39
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TP53 P04637 2/20 0.36
KMT2A Q03164 1/20 0.36
CASR P41180 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
ADRB2 P07550 1/20 0.35
IDO1 P14902 1/20 0.34
SLC6A9 P48067 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33
PDE2A O00408 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7780432 0.86 ALDH1A1 (0.41) ALDH1A1CYP3A4GAALMNATDP1
SCHEMBL7785127 0.86 ALDH1A1 (0.41) ALDH1A1CYP3A4GAALMNATDP1
SCHEMBL7780640 0.86 ALDH1A1 (0.41) ALDH1A1CYP3A4GAALMNATDP1
SCHEMBL7780398 0.82 TDP1 (0.46) ALDH1A1LMNAAKR1C3AKR1C2TDP1
SCHEMBL7787461 0.80 TDP1 (0.55) ALDH1A1CYP3A4GAALMNATDP1
SCHEMBL7789250 0.79 ALDH1A1 (0.41) ALDH1A1CYP3A4GAALMNAAKR1C3
SCHEMBL7780717 0.79 ALDH1A1 (0.41) ALDH1A1CYP3A4GAALMNAAKR1C3
SCHEMBL7780395 0.77 MEN1 (0.42) ALDH1A1KMT2ASLC6A9SLC6A5
Hydrochloric Acid SCHEMBL7785515 0.77 CXCR2 (0.43) ALDH1A1GAALMNAAKR1C3AKR1C2
SCHEMBL7784989 0.76 ACP3 (0.45) ALDH1A1CYP3A4AOC3GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed