SCHEMBL7780979

SCHEMBL7780979

Fc1cc(Oc2cccc(C(F)(F)F)c2)ncn1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
POLB P06746 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MAPT P10636 2/20 0.50
KDR P35968 8/20 0.47
MAPK14 Q16539 7/20 0.46
TNNI3K Q59H18 7/20 0.46
BRAF P15056 6/20 0.46
GAA P10253 1/20 0.44
MAPK1 P28482 1/20 0.44
TTBK1 Q5TCY1 1/20 0.44
LRRK2 Q5S007 1/20 0.43
TEAD1 P28347 1/20 0.43
TRPV1 Q8NER1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4244096 0.91 L3MBTL1 (0.57) ALDH1A1POLBL3MBTL1MAPTKDR
SCHEMBL12825474 0.84 KDR (0.62) ALDH1A1POLBL3MBTL1MAPTKDR
SCHEMBL16202045 0.84 KDR (0.62) ALDH1A1POLBL3MBTL1MAPTKDR
SCHEMBL7783065 0.84 ALDH1A1 (0.54) ALDH1A1POLBL3MBTL1MAPTKDR
SCHEMBL8773803 0.82 ALDH1A1 (0.53) ALDH1A1POLBL3MBTL1MAPTKDR
SCHEMBL8683754 0.82 ALDH1A1 (0.47) ALDH1A1POLBL3MBTL1MAPTKDR
SCHEMBL8941516 0.81 MAPT (0.59) ALDH1A1POLBL3MBTL1MAPTGAA
SCHEMBL8773158 0.80 MAPT (0.65) ALDH1A1POLBL3MBTL1MAPTGAA
SCHEMBL29607042 0.80 MAPT (0.65) ALDH1A1POLBL3MBTL1MAPTGAA
SCHEMBL7775883 0.79 MAPT (0.48) ALDH1A1POLBL3MBTL1MAPTKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0794177-B1 Process for the preparation of unsymmertical 4,6-Bis (aryloxy pyrimidine compounds AMERICAN CYANAMID CO (US) 2001-10-10 EP disclosed
US-6087498-A Process for the preparation of unsymmetrical 4,6-bis(aryloxy) pyrimidine compounds AMERICAN CYANAMID COMPANY (US) 2000-07-11 US disclosed
US-5977363-A Process for the preparation of unsymmetrical 4,6-bis(aryloxy) pyrimidine compounds AMERICAN CYANAMID COMPANY (US) 1999-11-02 US disclosed
EP-0794177-A1 Process for the preparation of unsymmertical 4,6-Bis (aryloxy pyrimidine compounds American Cyanamid Company (US) 1997-09-10 EP disclosed