SCHEMBL7781773

SCHEMBL7781773

CC(C)(C)OC(=O)NC1CCCCc2cc(OCC3CCCC(C(N)=O)C3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
SCN3A Q9NY46 1/20 0.38
PARP10 Q53GL7 5/20 0.38
PARP15 Q460N3 4/20 0.38
SRC P12931 4/20 0.38
ACACB O00763 1/20 0.38
BDKRB1 P46663 2/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
PARP2 Q9UGN5 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7659131 0.88 PARP10 (0.43) TAS1R3TAS1R1TAS1R2SCN3APARP10
SCHEMBL7654129 0.76 SRC (0.58) PARP10PARP15SRC
SCHEMBL7654125 0.76 SRC (0.58) PARP10PARP15SRC
SCHEMBL20533142 0.74 DRD2 (0.41) TAS1R3TAS1R1TAS1R2BDKRB1CA12
SCHEMBL20533140 0.74 DRD2 (0.41) TAS1R3TAS1R1TAS1R2BDKRB1CA12
SCHEMBL20683057 0.74 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2BDKRB1
SCHEMBL26073271 0.74 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2BDKRB1
SCHEMBL3537138 0.73 CFD (0.49) TAS1R3TAS1R1TAS1R2BDKRB1ALDH1A1
SCHEMBL3537141 0.73 CFD (0.49) TAS1R3TAS1R1TAS1R2BDKRB1ALDH1A1
SCHEMBL16809810 0.73 KMT2A (0.44) TAS1R3TAS1R1TAS1R2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129068-A1 BICYCLIC SIGNAL TRANSDUCTION INHIBITORS, COMPOSITION CONTAINING THEM AND USES THEREOF ARIAD PHARMACEUTICALS, INC. (US) 2001-09-05 EP disclosed
WO-2000027802-A1 BICYCLIC SIGNAL TRANSDUCTION INHIBITORS, COMPOSITIONS CONTAINING THEM & USES THEREOF ARIAD PHARMACEUTICALS, INC. (US) 2000-05-18 WO disclosed