SCHEMBL7783101

SCHEMBL7783101

CC(=O)C(N)c1ccc(Cl)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.44
ALDH1A1 P00352 1/20 0.44
BRD4 O60885 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
DGAT1 O75907 1/20 0.38
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 1/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
EPHX1 P07099 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13049949 0.85 NAPRT (0.48) NAPRTALDH1A1CYP3A4CYP2D6SLC6A2
SCHEMBL13235872 0.81 NAPRT (0.44) NAPRTALDH1A1BRD4CYP3A4CYP2D6
SCHEMBL27672314 0.79 LMNA (0.48) NAPRTALDH1A1CYP3A4CYP2D6DGAT1
SCHEMBL890206 0.77 ALDH1A1 (0.41) NAPRTALDH1A1BRD4CYP3A4CYP2D6
SCHEMBL594241 0.76 ADRB2 (0.52) NAPRTCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL19943572 0.76 CYP3A4 (0.45) NAPRTALDH1A1CYP3A4CYP2D6SLC6A2
SCHEMBL31247543 0.76 ADRB2 (0.52) NAPRTCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL4092765 0.76 ADRB2 (0.52) NAPRTCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL31086606 0.76 ADRB2 (0.52) NAPRTCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL14211414 0.76 ADRB2 (0.52) NAPRTCYP3A4CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691331-B1 Process for the preparation of n-acylated 2-chloro-5-aminomethyl-pyridines BAYER AG (DE) 2001-10-10 EP disclosed
US-5580983-A Process for the preparation of N-acylated 2-chloro-5-aminomethylpyridines BAYER AKTIENGESELLSCHAFT (DE) 1996-12-03 US disclosed
EP-0691331-A1 Process for the preparation of n-acylated 2-chloro-5-aminomethyl-pyridines BAYER AG (DE) 1996-01-10 EP disclosed