SCHEMBL7783271

SCHEMBL7783271

CC(N)c1ccc(-c2ccccc2)cc1.CC(N)c1ccc(F)c(C(F)(F)F)c1.NCCc1ccc(Cl)c(C(F)(F)F)c1.NCCc1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 8/20 0.39
TAAR1 Q96RJ0 2/20 0.38
TP53 P04637 1/20 0.37
IDO1 P14902 2/20 0.35
SLC6A3 Q01959 3/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
MMP7 P09237 1/20 0.34
RPS6KB1 P23443 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846362 0.98 MAOB (0.40) MAOBTAAR1TP53IDO1SLC6A3
SCHEMBL7782593 0.90 IDO1 (0.42) MAOBTAAR1IDO1SLC6A3
SCHEMBL7865721 0.84 TAAR1 (0.45) MAOBTAAR1RPS6KB1
SCHEMBL7846359 0.83 TP53 (0.43) TP53SLC6A3AKR1C3AKR1C2
SCHEMBL7782591 0.82 ADRB2 (0.42) TP53IDO1SLC6A3AKR1C3AKR1C2
Ammonia Solution, Strong SCHEMBL7569458 0.82 IDO1 (0.40) IDO1SLC6A3
SCHEMBL7865718 0.75 PDE2A (0.42) AKR1C3AKR1C2RPS6KB1
SCHEMBL27220940 0.71 TAAR1 (0.50) MAOBTAAR1
SCHEMBL13877352 0.71 ADRB2 (0.45) IDO1AKR1C3AKR1C2
SCHEMBL27687280 0.71 IDO1 (0.62) MAOBTAAR1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144397-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144397-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034258-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed