SCHEMBL7784038

SCHEMBL7784038

C=CCNC(=O)C1CNCC[N]1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 1/20 0.35
TSHR P16473 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787553 0.80 KMT2A (0.34) KMT2A
SCHEMBL7786231 0.76 CHRNB2 (0.47) KMT2AKDM4EALDH1A1MEN1
SCHEMBL1834987 0.76
SCHEMBL752438 0.73 CHRNB2 (0.40)
SCHEMBL2301489 0.72 KMT2A (0.70) KMT2ANPSR1LMNATSHRSMN1; SMN2
SCHEMBL7765233 0.71 KMT2A (0.49) KMT2ANPSR1LMNATSHRSMN1; SMN2
SCHEMBL4984 0.69 CHRNB2 (0.40)
SCHEMBL5661852 0.69 CHRNB2 (0.44) KMT2ASMN1; SMN2MEN1
SCHEMBL9053082 0.69 L3MBTL1 (0.36) ALDH1A1
SCHEMBL2915925 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866609-A PROPHYLACTIC AND THERAPEUTIC AGENTS FOR ARTERIOSCLEROSIS. SS PHARMACEUTICAL CO., LTD. (JP) 1999-02-02 US claimed
EP-0823420-A2 Substituted vinylurea derivatives and their use as ACAT inhibitors SS PHARMACEUTICAL CO., LTD. (JP) 1998-02-11 EP claimed
EP-0823420-B1 Substituted vinylurea derivatives and their use as ACAT inhibitors SS PHARMACEUTICAL CO (JP) 2001-10-24 EP disclosed
US-5866609-A PROPHYLACTIC AND THERAPEUTIC AGENTS FOR ARTERIOSCLEROSIS. SS PHARMACEUTICAL CO., LTD. (JP) 1999-02-02 US disclosed
EP-0823420-A2 Substituted vinylurea derivatives and their use as ACAT inhibitors SS PHARMACEUTICAL CO., LTD. (JP) 1998-02-11 EP disclosed