SCHEMBL7784865

SCHEMBL7784865

O=C(O)c1ccc2c(CCCCN3CCN(c4cc(=O)oc5cc(F)ccc45)CC3)c[nH]c2c1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.49
DRD2 P14416 1/20 0.49
HTR7 P34969 2/20 0.46
ADRA1A P35348 1/20 0.46
KCNH2 Q12809 1/20 0.46
MPO P05164 1/20 0.46
SLC6A4 P31645 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203156 0.94 HTR1A (0.54) HTR1AHTR7ADRA1AKCNH2MPO
SCHEMBL8133408 0.93 HTR1A (0.50) HTR1ADRD2HTR7ADRA1AKCNH2
SCHEMBL7787382 0.91 HTR1A (0.47) HTR1ADRD2HTR7ADRA1AKCNH2
SCHEMBL7784880 0.90 HTR1A (0.44) HTR1ADRD2ADRA1A
SCHEMBL7780263 0.90 DRD2 (0.49) HTR1ADRD2KCNH2SLC6A4
SCHEMBL7787373 0.90 KDM4E (0.47) HTR1ADRD2
SCHEMBL7787585 0.88 HTR1A (0.51) HTR1ADRD2HTR7ADRA1AKCNH2
SCHEMBL7784858 0.88 ADRA2A (0.53) HTR1ADRD2ADRA1A
SCHEMBL7787379 0.85 DRD2 (0.57) HTR1ADRD2HTR7ADRA1AKCNH2
SCHEMBL7780259 0.85 SLC6A4 (0.53) HTR1AHTR7ADRA1AKCNH2MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1093127-C Piperazine derivatives MERCK PATENT GMBH (DE) 2002-10-23 CN disclosed
US-6251908-B1 Piperazine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2001-06-26 US disclosed
CN-1264379-A Piperazine derivatives MERCK PATENT GMBH (DE) 2000-08-23 CN disclosed