SCHEMBL7784886

SCHEMBL7784886

N#Cc1ccc2c(CCCCN3CCN(c4cc(=O)oc5ccccc45)CC3)c[nH]c2c1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.55
DRD2 P14416 1/20 0.55
HTR2A P28223 1/20 0.55
HTR6 P50406 1/20 0.52
KCNH2 Q12809 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201581 0.93 HTR1A (0.63) HTR1ADRD2HTR2AHTR6KCNH2
SCHEMBL7787397 0.88 HTR1A (0.59) HTR1ADRD2
SCHEMBL7787379 0.87 DRD2 (0.57) HTR1ADRD2KCNH2
SCHEMBL7784884 0.87 DRD2 (0.57) HTR1ADRD2HTR6KCNH2
SCHEMBL7787585 0.86 HTR1A (0.51) HTR1ADRD2HTR2AHTR6KCNH2
SCHEMBL7787373 0.85 KDM4E (0.47) HTR1ADRD2
SCHEMBL7788889 0.85 HTR1A (0.57) HTR1ADRD2HTR2A
SCHEMBL7784868 0.84 HTR1A (0.49) HTR1ADRD2HTR6KCNH2
SCHEMBL7787574 0.83 HTR1A (0.48) HTR1ADRD2KCNH2
SCHEMBL8131459 0.83 DRD2 (0.46) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1093127-C Piperazine derivatives MERCK PATENT GMBH (DE) 2002-10-23 CN disclosed
US-6251908-B1 Piperazine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2001-06-26 US disclosed
EP-0998474-A1 PIPERAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2000-05-10 EP disclosed
WO-1999003855-A1 PIPERAZINE DERIVATIVES MERCK PATENT GMBH (DE) 1999-01-28 WO disclosed