SCHEMBL7785101

SCHEMBL7785101

C[C@@H](NC(c1ccc(Cl)cc1)c1cccc(N)c1)c1ccc(F)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.36
AKT1 P31749 2/20 0.35
CYP3A4 P08684 4/20 0.35
CYP2D6 P10635 4/20 0.35
SLC6A2 P23975 4/20 0.35
SLC6A4 P31645 4/20 0.35
SLC6A3 Q01959 4/20 0.35
KCNH2 Q12809 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPKAPK2 P49137 1/20 0.34
S1PR1 P21453 2/20 0.33
S1PR3 Q99500 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PDPK1 O15530 1/20 0.33
SCN1A P35498 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN8A Q9UQD0 1/20 0.32
LDHA P00338 1/20 0.32
LDHB P07195 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7784936 0.92 PDPK1 (0.39) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL27553525 0.92 PDPK1 (0.39) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7789259 0.91 ADRB2 (0.35) ADRB2AKT1CYP3A4CYP2D6SLC6A2
SCHEMBL7785573 0.91 ADRB2 (0.35) ADRB2AKT1CYP3A4CYP2D6SLC6A2
SCHEMBL7780509 0.91 MAPKAPK2 (0.34) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7785234 0.91 MAPKAPK2 (0.34) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7780705 0.90 LMNA (0.34) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7785653 0.90 SLC6A2 (0.36) ADRB2AKT1CYP3A4CYP2D6SLC6A2
SCHEMBL7785553 0.90 LMNA (0.34) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7787609 0.88 MAPKAPK2 (0.45) AKT1KMT2AMAPKAPK2ALDH1A1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed