SCHEMBL7787609

SCHEMBL7787609

CC(NC(c1ccncc1)c1cccc(N)c1)c1ccc(F)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.45
AKT1 P31749 2/20 0.36
TRPV1 Q8NER1 1/20 0.33
KRAS P01116 1/20 0.33
SOS1 Q07889 1/20 0.33
MAPK1 P28482 2/20 0.32
RPS6KB1 P23443 2/20 0.32
ROCK1 Q13464 2/20 0.32
RPS6KA5 O75582 1/20 0.32
MAP4K4 O95819 1/20 0.32
PRKCG P05129 1/20 0.32
CDK1 P06493 1/20 0.32
PRKACA P17612 1/20 0.32
CDK2 P24941 1/20 0.32
AKT2 P31751 1/20 0.32
FLT4 P35916 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
IRAK1 P51617 1/20 0.32
RPS6KA3 P51812 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27553525 0.90 PDPK1 (0.39) MAPKAPK2KRASSOS1MAPK1RPS6KB1
SCHEMBL7784936 0.90 PDPK1 (0.39) MAPKAPK2KRASSOS1MAPK1RPS6KB1
SCHEMBL7785234 0.89 MAPKAPK2 (0.34) MAPKAPK2KRASSOS1MAPK1RPS6KB1
SCHEMBL7780509 0.89 MAPKAPK2 (0.34) MAPKAPK2KRASSOS1MAPK1RPS6KB1
SCHEMBL7785553 0.88 LMNA (0.34) MAPKAPK2KRASSOS1MAPK1RPS6KB1
SCHEMBL7780705 0.88 LMNA (0.34) MAPKAPK2KRASSOS1MAPK1RPS6KB1
SCHEMBL7785101 0.88 ADRB2 (0.36) MAPKAPK2AKT1KRASSOS1MAPK1
SCHEMBL7785301 0.84 MAPKAPK2 (0.47) MAPKAPK2AKT1MAPK1RPS6KB1ROCK1
SCHEMBL7780640 0.84 ALDH1A1 (0.41) KRASSOS1MAPTGAAALDH1A1
SCHEMBL7780432 0.84 ALDH1A1 (0.41) KRASSOS1MAPTGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed