SCHEMBL7785652

SCHEMBL7785652

CN(C)CC#Cc1ccc(C#N)cc1.CN(C)CC#Cc1ccc([N+](=O)[O-])cc1.COc1ccc(C#CCN(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
LMNA P02545 2/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 6/20 0.43
NPC1 O15118 2/20 0.43
PKM P14618 1/20 0.43
GAA P10253 1/20 0.43
CYP19A1 P11511 2/20 0.43
APP P05067 1/20 0.42
KCNH2 Q12809 3/20 0.41
KCNJ1 P48048 2/20 0.41
RAB9A P51151 2/20 0.40
MEN1 O00255 1/20 0.39
MITF O75030 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378545 0.84 PYCR1 (0.46) ALDH1A1POLBMAPTGAAKCNH2
SCHEMBL7081483 0.80 APP (0.50) APPKCNH2
SCHEMBL4508653 0.78 APP (0.58) ALDH1A1LMNAPOLBMAPTNPC1
SCHEMBL7080591 0.77 CYP2A6 (0.49) ALDH1A1CYP19A1KCNH2
SCHEMBL27214761 0.73 KCNJ1 (0.55) ALDH1A1LMNAMAPTNPC1PKM
SCHEMBL3128583 0.72 HSPB1 (0.59) ALDH1A1LMNAPOLBMAPTNPC1
Nitrogen SCHEMBL9082924 0.72 APP (0.66) ALDH1A1LMNAPOLBMAPTNPC1
SCHEMBL57257 0.72 VCAM1 (0.61) ALDH1A1LMNAMAPTNPC1PKM
SCHEMBL492221 0.72 APP (0.70) ALDH1A1LMNAPOLBMAPTNPC1
SCHEMBL20328414 0.72 APP (0.70) ALDH1A1LMNAPOLBMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137633-A2 ACETAMIDE AND SUBSTITUTED ACETAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
WO-2000034237-A2 ACETAMIDE AND SUBSTITUTED ACETAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed