SCHEMBL7787455

SCHEMBL7787455

COc1ccc(C(NC(C)c2ccc(F)c(F)c2)c2cc(N)ccc2OC)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.39
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
ACHE P22303 3/20 0.38
HTT P42858 2/20 0.36
ADRA2A P08913 2/20 0.35
ADRA1A P35348 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPK1 P28482 2/20 0.34
MEN1 O00255 1/20 0.34
BLM P54132 1/20 0.34
KMT2A Q03164 1/20 0.34
CHRM4 P08173 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7780363 0.92 CA1 (0.34) CYP2D6CA1CA2ACHEALDH1A1
SCHEMBL7784903 0.92 ALDH1A1 (0.37) CA1CA2ACHEHTTALDH1A1
SCHEMBL7787479 0.89 MEN1 (0.39) CYP2D6CA1CA2ACHEALDH1A1
SCHEMBL7780319 0.87 CYP2D6 (0.40) CYP2D6CA1CA2ACHEHTT
SCHEMBL7780785 0.87 TDP1 (0.43) CA1CA2ACHEHTTALDH1A1
SCHEMBL7780568 0.84 ALDH1A1 (0.39) CA1CA2ACHEHTTALDH1A1
SCHEMBL7785707 0.82 MAPT (0.43) HTTALDH1A1MAPTL3MBTL1MAPK1
SCHEMBL7780640 0.81 ALDH1A1 (0.41) CA1CA2ACHEHTTALDH1A1
SCHEMBL7780432 0.81 ALDH1A1 (0.41) CA1CA2ACHEHTTALDH1A1
SCHEMBL7785127 0.81 ALDH1A1 (0.41) CA1CA2ACHEHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed