SCHEMBL7789426

SCHEMBL7789426

COc1ccc(C(NC(=O)c2cccc(F)c2)c2cccc([N+](=O)[O-])c2)cc1

nearest known ligand 0.74

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.74
LMNA P02545 3/20 0.74
GAA P10253 2/20 0.74
MAPT P10636 2/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
KDM4E B2RXH2 1/20 0.52
TP53 P04637 2/20 0.52
KMT2A Q03164 2/20 0.52
CYP3A4 P08684 1/20 0.49
MEN1 O00255 1/20 0.48
GPR17 Q13304 2/20 0.47
P2RY2 P41231 1/20 0.47
HTT P42858 1/20 0.47
SLC6A9 P48067 1/20 0.45
SLC6A5 Q9Y345 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7780334 0.91 ALDH1A1 (0.70) ALDH1A1LMNAGAAMAPTNPC1
SCHEMBL7785221 0.89 ALDH1A1 (0.64) ALDH1A1LMNAGAAMAPTNPC1
SCHEMBL7785664 0.83 ALDH1A1 (0.56) ALDH1A1LMNAGAAMAPTNPC1
Hydrochloric Acid SCHEMBL7785398 0.82 ALDH1A1 (0.79) ALDH1A1LMNAGAANPC1RAB9A
SCHEMBL7780405 0.82 LMNA (0.48) ALDH1A1LMNAGAAMAPTNPC1
SCHEMBL7780373 0.82 LMNA (0.48) ALDH1A1LMNAGAAMAPTNPC1
SCHEMBL27530409 0.79 MAPK1 (0.47) ALDH1A1LMNAGAAMAPTNPC1
SCHEMBL7785483 0.79 MAPK1 (0.47) ALDH1A1LMNAGAAMAPTNPC1
SCHEMBL12350147 0.79 MEN1 (0.54) ALDH1A1LMNAMAPTNPC1RAB9A
SCHEMBL10155639 0.78 MAPT (0.47) ALDH1A1LMNAGAAMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed